Cholinesterase Research
| Cholinesterase Research |
| Autore | Korabecny Jan |
| Pubbl/distr/stampa | Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021 |
| Descrizione fisica | 1 online resource (223 p.) |
| Soggetto topico | Medicine and Nursing |
| Soggetto non controllato |
acetylcholinesterase
acetylcholinesterase inhibitor acetylcholinesterase inhibitors alkaloids Alzheimer disease Alzheimer's disease Amaryllidaceae antioxidants behavior blood-brain barrier crossing bone healing butyrylcholinesterase butyrylcholinesterase inhibitors carltonine A-C catalysis cholinesterase dementia docking docking studies donepezil fluorene hemostasis hydrolysis in silico in vitro inhibition MD simulations molecular dynamics molecular modeling molecular modelling molecular recognition multi-target directed ligands N-methyl-d-aspartate receptor n/a Narcissus pseudonarcissus cv. Carlton neutron scattering nutraceuticals organophosphates organophosphorus organophosphorus nerve agents osmotic stress osseointegration oxime pharmacodynamics phytochemicals reactivation reactivation process reactivators slow-binding inhibition transition state analog ventilation zebrafish |
| Formato | Materiale a stampa |
| Livello bibliografico | Monografia |
| Lingua di pubblicazione | eng |
| Record Nr. | UNINA-9910557764703321 |
Korabecny Jan
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| Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021 | ||
| Lo trovi qui: Univ. Federico II | ||
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Computational Approaches: Drug Discovery and Design in Medicinal Chemistry and Bioinformatics
| Computational Approaches: Drug Discovery and Design in Medicinal Chemistry and Bioinformatics |
| Autore | Tutone Marco |
| Pubbl/distr/stampa | Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021 |
| Descrizione fisica | 1 online resource (387 p.) |
| Soggetto topico |
Chemistry
Research & information: general |
| Soggetto non controllato |
3CL-Pro
3D-QSAR acetylcholinesterase aging progression mechanism Alzheimer's disease aminophenylbenzamide antibody:antigen interactions antivirals binding free energies binding site binding space carbon nanotubes cholesterol computational biology consensus models COVID-19 COX-2 inhibitors deep learning diabetes docking simulations doxorubicin encapsulation drug delivery system drug discovery drug repositioning drug repositioning approaches drug repurposing drug resistance drug-resistance mutations dual mode of action dual-target lead discovery epitope binning epitope mapping epitope prediction FimH fingerprints gene expression signature genome-wide genetic and epigenetic network (GWGEN) glycoprotein D (gD) haeckelite defects HDACs hERG toxicity herpes simplex virus fusion proteins high-throughput virtual screening HIV-2 protease homology modeling hTSPO human dihydrofolate reductase immunoproteasome in silico induced structural deformations induced-fit docking inhibitors isoform-selective histone deacetylase inhibitors isomeric space ligand-based model machine learning main protease MD binding MD simulation metadynamics methotrexate molecular docking molecular dynamics molecular dynamics (MD) simulation molecular dynamics simulation molecular dynamics simulations molecular modeling MRP4 multi-modal multiple-molecule drug multiprotein inhibiting natural compounds multiscale multitargeting mutants Mycobacterium tuberculosis n/a natural compounds neurodegenerative disorders nicotinic acetylcholine receptor non-covalent inhibitors noncovalent interactions oxidative stress PF-00835231 pharmacophore model pharmacophore modeling PK11195 polypharmacology proteasome protein docking protein threading modeling proteomic signature RNA expression regulation SARS-CoV-2 skin aging SNPs sodium-glucose co-transporters 2 Src inhibitors Stone-Wales defects structural bioinformatics structural characterization systems medicine design tuberculosis urinary tract infections uropathogenic bacteria variants virtual screening |
| Formato | Materiale a stampa |
| Livello bibliografico | Monografia |
| Lingua di pubblicazione | eng |
| Altri titoli varianti | Computational Approaches |
| Record Nr. | UNINA-9910557519403321 |
Tutone Marco
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| Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021 | ||
| Lo trovi qui: Univ. Federico II | ||
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Drug-Drug Interactions
| Drug-Drug Interactions |
| Autore | Kim Dong Hyun |
| Pubbl/distr/stampa | Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021 |
| Descrizione fisica | 1 online resource (242 p.) |
| Soggetto topico |
Biology, life sciences
Research & information: general |
| Soggetto non controllato |
(‒)-sophoranone
1A2 2B6 2C19 2C8 2C9 2D6 3A4 ADME adverse drug reactions biflavonoid chronic kidney disease competitive inhibition computational prediction CYP CYP1A1 CYP1A2 CYP2C9 CYP2D6 CYP3A CYP3A4 cytochrome P450 cytochromes P450 DDI Dexamethasone drug interaction drug interactions drug metabolism drug transporter drug-drug interaction drug-drug interactions expression fexofenadine gepants high plasma protein binding in silico in vitro in vivo inhibitor ixazomib Ketoconazole lasmiditan Lexicomp low permeability Loxoprofen mechanism-based inhibition metabolic DDI metabolism migraine monoclonal antibodies non-competitive inhibition O-desmethyltramadol OATP1B1 OATP1B3 organic anion transporting polypeptide 1A2 (OATP1A2) P-glycoprotein (P-gp) P450 pharmacokinetics physiologically-based pharmacokinetics plasma concentration polypharmacy potent inhibition QSAR regulation Rumex acetosa selamariscina A signal detection algorithms spontaneous reporting systems subset analysis substrate systemic exposure tadalafil ticagrelor tissue-specific tramadol tyrosine kinase inhibitors ubiquitination uridine 5'-diphosphoglucuronosyl transferase |
| Formato | Materiale a stampa |
| Livello bibliografico | Monografia |
| Lingua di pubblicazione | eng |
| Record Nr. | UNINA-9910557666403321 |
Kim Dong Hyun
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| Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021 | ||
| Lo trovi qui: Univ. Federico II | ||
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From a Molecule to a Drug: Chemical Features Enhancing Pharmacological Potential
| From a Molecule to a Drug: Chemical Features Enhancing Pharmacological Potential |
| Autore | Ribaudo Giovanni |
| Pubbl/distr/stampa | Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022 |
| Descrizione fisica | 1 online resource (234 p.) |
| Soggetto topico |
Medicine and Nursing
Pharmacology |
| Soggetto non controllato |
3-chymotrypsin-like protease
affinity chromatography alginate anti-ACE anti-DPP-IV anti-inflammatory drugs antioxidant activity benzoic acid derivatives big data binding free energy Box-Behken breast milk cannabinoid chemoinformatics chromatographic descriptors cisplatin clopidogrel coronavirus SARS-CoV-2 COVID-19 cyclooxygenase cytoprotection DFT calculations drug compounding drug discovery E-selectin Eucheuma gelatinae extraction fucoidan gallic acid gastrointestinal digestion high performance liquid chromatography ICAM-1 imine-enamine in silico L-selectin lithium therapy M/P ratio MCP-1 methadone hydrochloride microbiology molecular descriptors molecular docking molecular dynamics molecular dynamics simulations monocyte migration multitarget drug n/a nephrotoxicity neurocytology neuropathic pain neuroprotection NMR study one-pot oxone pain management paramyosin peroxymonosulfate pharmaceutical solutions pharmacodynamics pharmacokinetics physic-chemistry precision medicine protein binding pyrimidonic pharmaceuticals QSAR quercetin quercetin 3-O-glucuronide reaction mechanism reactivity parameters rheology SARS-CoV-2 seafood selenium selenoxide elimination sodium halide stability study statistical modeling target fishing thienopyridine THP-1 macrophage toxicology β-carrageenan |
| Formato | Materiale a stampa |
| Livello bibliografico | Monografia |
| Lingua di pubblicazione | eng |
| Altri titoli varianti | From a Molecule to a Drug |
| Record Nr. | UNINA-9910585940503321 |
Ribaudo Giovanni
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| Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022 | ||
| Lo trovi qui: Univ. Federico II | ||
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Metabolomics Data Processing and Data Analysis-Current Best Practices
| Metabolomics Data Processing and Data Analysis-Current Best Practices |
| Autore | Hanhineva Kati |
| Pubbl/distr/stampa | Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021 |
| Descrizione fisica | 1 online resource (276 p.) |
| Soggetto topico | Research & information: general |
| Soggetto non controllato |
all ion fragmentation
biostatistics bootstrapped-VIP chemical classification combinatorial fragmentation compound identification computational metabolomics computational statistical constraint-based modeling data processing data repository data-dependent acquisition (DDA) data-independent acquisition disease risk enrichment analysis environmental factors experimental design flux balance forensics fragmentation (MS/MS) full-scan MS/MS processing genome-scale metabolic modeling global metabolomics gut microbiome host-microbiome in silico in silico workflows ion selection algorithms LC-MS lipidomics liquid chromatography liquid chromatography high-resolution mass spectrometry liquid chromatography mass spectrometry liquid chromatography-mass spectrometry (LC-MS) liquid chromatography-mass spectrometry (LC/MS) mass spectral libraries mass spectrometry mass spectrometry imaging meta-omics metabolic networks metabolic pathway and network analysis metabolic profiling metabolic reconstructions metabolism metabolite annotation metabolite identification metabolome mining metabolomics metabolomics data mapping metabolomics imaging metagenomics molecular families MS spectral prediction multivariate risk modeling networking nontarget analysis NPLS pathway analysis PLS R programming R-MetaboList 2 reanalysis rule-based fragmentation sample preparation simulator spectra processing structure-based chemical classification substructures supervised learning tandem mass spectral library targeted analysis time series triplot univariate and multivariate statistics unsupervised learning untargeted analysis untargeted metabolomics variable selection wastewater |
| Formato | Materiale a stampa |
| Livello bibliografico | Monografia |
| Lingua di pubblicazione | eng |
| Record Nr. | UNINA-9910557354403321 |
Hanhineva Kati
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| Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021 | ||
| Lo trovi qui: Univ. Federico II | ||
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Molecular Computing and Bioinformatics / Xiangxiang Zeng, Quan Zou, Alfonso Rodríguez-Patón
| Molecular Computing and Bioinformatics / Xiangxiang Zeng, Quan Zou, Alfonso Rodríguez-Patón |
| Autore | Zeng Xiangxiang |
| Pubbl/distr/stampa | MDPI - Multidisciplinary Digital Publishing Institute, 2019 |
| Descrizione fisica | 1 electronic resource (390 p.) |
| Soggetto topico | Biotechnology |
| Soggetto non controllato |
systems biology
join graph hierarchical support vector regression transcription factor brain storm optimization heterogeneous information network embedding structural patterns gene fusion data Panax ginseng flowering plant geometric arithmetic index interspecies transmission iron-depleted drug discovery protein protein targeting recursively enumerable function Mycoplasma hominis environmental factor Alzheimer’s disease absorption angiogenesis classification self-organizing systems enzymatic numerical P system excretion atom-bond connectivity index molecular learning DNA coding phylogeny bone formation DCL1 line graph pseudo dinucleotide composition load balancing K2 efflux ratio osteogenesis distribution NanoString Technologies RAST server 8-bit adder/subtractor gene networks dihydrouridine structure information Cartesian product graph domain label stacking denoising auto-encoder DNA computing Stenotrophomonas maltophilia pattern classification stress causal direction learning machine learning adverse drug reaction prediction membrane computing support vector machine Brassica napus miRNA biogenesis identification of Chinese herbal medicines bio-inspired toxicity protein transduction domain RNA sequence information multiple interaction networks in silico protein complex drug low-dimensional representation gene coding protein amino acid mutation Bayesian causal model edge detection big data function prediction parallel computing resolution free Hamming distance cascade oligopeptide transporter DNA barcoding technology DNA strand displacement protein–protein interaction (PPI) biomedical text mining bioinformatics metabolism hypoxia-inducible factor-1? nucleotide physicochemical property Turing universality diabetes mellitus chaotic map multinetwork integration bacterial computing lignification penalized matrix decomposition ensemble classifier bacteria and plasmid system similarity network RNA secondary structure avian influenza virus evaluating driver partner image encryption siderophores meta-path-based proximity P-glycoprotein Tianhe-2 prostate cancer iron acquisition systems biochip technology gene susceptibility prioritization laccase DNA molecular computing microRNA clustering drug-target interaction prediction endoplasmic reticulum |
| ISBN |
9783039211968
303921196X |
| Formato | Materiale a stampa |
| Livello bibliografico | Monografia |
| Lingua di pubblicazione | eng |
| Record Nr. | UNINA-9910346836303321 |
Zeng Xiangxiang
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| MDPI - Multidisciplinary Digital Publishing Institute, 2019 | ||
| Lo trovi qui: Univ. Federico II | ||
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New Advances in the Research of Antioxidant Food Peptides
| New Advances in the Research of Antioxidant Food Peptides |
| Autore | Amigo Lourdes |
| Pubbl/distr/stampa | Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021 |
| Descrizione fisica | 1 online resource (154 p.) |
| Soggetto topico | Research and information: general |
| Soggetto non controllato |
aged animals
albumin albumin peptide animal protein antioxidant antioxidant activity antioxidant enzymes antioxidant peptide antioxidant peptides bioactive peptide bioactive peptides C2C12 cell models cellular ROS egg white egg yolk exercise extraction food antioxidant food peptides fruit residues HepG2 hydrolysis condition in silico multifunctionality mung bean mung bean albumin muscle n/a older adult ORAC peptide sequencing peptides reactive oxygen species sarcopenia Vigna radiata whey protein whey protein hydrolysate |
| Formato | Materiale a stampa |
| Livello bibliografico | Monografia |
| Lingua di pubblicazione | eng |
| Record Nr. | UNINA-9910557793003321 |
Amigo Lourdes
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| Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021 | ||
| Lo trovi qui: Univ. Federico II | ||
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New Biomolecules and Drug Delivery Systems as Alternatives to Conventional Antibiotics
| New Biomolecules and Drug Delivery Systems as Alternatives to Conventional Antibiotics |
| Autore | Felgueiras Helena |
| Pubbl/distr/stampa | Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022 |
| Descrizione fisica | 1 online resource (232 p.) |
| Soggetto topico |
Chemistry
Research & information: general |
| Soggetto non controllato |
4-Nerolidylcatechol
aerosol delivery allicin antibacterial activity antibiotic antibiotic discovery antibiotics antifungals antimicrobial activity Azadirachta indica biodegradable polymers biofilm bone regeneration and nanofiber scaffold bulk-tank milk Catharanthus roseus chitosan colistin biosynthetic gene cluster controlled release conventional antibiotics cyclic diphenylphosphonate DNA gyrase DNA gyrase inhibitor drug delivery platforms efficient promoters fiber-hydrogel composite flavonoids goat gold nanoparticles Gram-negative bacteria gram-negative pathogens grapefruit seed extract green synthesis method hypertonic saline in silico kiwifruit disease live biosensors local prevention magnesium ion magnesium-doped calcium silicate mastitis methicillin microfluidic droplet cocultivation Microsporum canis milk molecular docking multi-omics multidrug-resistant Acinetobacter baumannii (MDR-AB) multidrug-resistant bacteria n/a nanoparticles nanoprecipitation nosocomial infection osteogenic activity plant extract polycaprolactone polymyxins prosthetic joint infection quercetin quinoline Rosa roxburghii silver nanoparticles single cell skin regeneration somatic cell counts Sphaerotheca sp staphylococcus storage quality tetracycline tetramycin total bacterial counts ultrahigh-throughput screening wound healing |
| Formato | Materiale a stampa |
| Livello bibliografico | Monografia |
| Lingua di pubblicazione | eng |
| Record Nr. | UNINA-9910585940303321 |
Felgueiras Helena
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| Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022 | ||
| Lo trovi qui: Univ. Federico II | ||
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Peptides for Health Benefits 2019 : Volume 1
| Peptides for Health Benefits 2019 : Volume 1 |
| Autore | Hernández-Ledesma Blanca |
| Pubbl/distr/stampa | Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2020 |
| Descrizione fisica | 1 online resource (340 p.) |
| Soggetto topico |
Biology, life sciences
Research & information: general |
| Soggetto non controllato |
ACE-inhibitory activity
acrylamide airway inflammation alcalase hydrolysate Alzheimer's disease AMD AMP identification and design amyloid amyloid fibrils and endothelial regeneration angiogenic precursor cells angiotensin I converting enzyme anti-biofilm peptides anti-inflammatory antibiotic resistance antifungal activity antigen-specific antihypertensive peptides antimicrobial peptide antimicrobial peptides antimicrobial peptides (AMPs) antimicrobial resistance antioxidant activity antioxidant peptide antiproliferative assay antisepsis, peptide antibiotics apolipoprotein E arthritis asthma Aβ peptide bioactive peptide bioactive peptides biomarkers BIOPEP-UWM database biosynthesis bone erosion cancer antigen cancer stem cells cartilage destruction cathelicidins Cec-analogs Cecropins central nervous system diseases chemoprevention Chlorella sorokiniana chronic diseases Clostridioides difficile CNV collagen collagen peptide colorectal cancer combinatorial library confocal microscopy conjugation copper Crassostrea angulata cryptides CXCR3 cystic fibrosis cytoprotective effect database defensins diseases docetaxel doxorubicin dry-cured pork ham dyslipidemia endothelial dysfunction endothelial progenitor cells energy expenditure enteric nervous system enzyme extra domain B fermentation fetal bovine serum (FBS) fibroblasts fibronectin Fmoc/tBu food intake regulation food-derived foods formyl peptide receptors FPYLRH fresh tissue functional food galanin gender differences glioma GPR10 Histatin-5 host defense peptides Hs02 human antimicrobial peptides human keratinocytes humanized mouse hybrid peptide hydrolysis hydroxyprolyl-glycine (Hyp-Gly) hyperglycemia hypertension immune checkpoint inhibitor immune response immune suppression immunomodulant in silico In situ tetramer staining inflammation inflammatory bowel disease insects intragenic antimicrobial peptide Lactoferricin B (Lfcin B) library design ligands lunasin MDA MDR infectious diseases membrane activity MHC tetramer migration miiuy croaker (Miichthys miiuy) mode of action molecular blind docking molecular docking molecular weight monocyte MRSA multimeric peptides mutagenesis n/a nano liquid chromatography tandem mass spectrometry (nanoLC-nanoESI MS/MS) neuroprotection neurotensin NF-κB non-atopic asthma nutraceuticals nutrition obesity oral delivery osteostatin oxidative stress pegylated glucagon-like peptide 1 peptide peptide vaccine peptide-drug conjugate physico-chemical properties PI3K/Akt pathway pidotimod pig piscidins platelets polymicrobial biofilms pro-inflammatory pro-inflammatory cytokines prolactin-releasing peptide prolyl-hydroxyproline (Pro-Hyp) prostate cancer protection ability proteolysis proteome microarray proteomics pseudin-2 Pseudomonas aeruginosa pulmonary emphysema RF-amide peptides rheumatic diseases screening sheepskin signaling Sjögren's syndrome SMILES code solid-phase synthesis sPLA2 Staphylococcus aureus stomach swim bladder synergistic effects synergy T cell T cells targeting temporin therapeutic potential type 1 diabetes vasoactive intestinal peptide VEGFR1 velvet antler VPAC1 receptor VPAC2 receptor whey peptides Αβ oligomer |
| Formato | Materiale a stampa |
| Livello bibliografico | Monografia |
| Lingua di pubblicazione | eng |
| Altri titoli varianti | Peptides for Health Benefits 2019 |
| Record Nr. | UNINA-9910557631703321 |
Hernández-Ledesma Blanca
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| Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2020 | ||
| Lo trovi qui: Univ. Federico II | ||
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Peptides for Health Benefits 2019 : Volume 2
| Peptides for Health Benefits 2019 : Volume 2 |
| Autore | Hernández-Ledesma Blanca |
| Pubbl/distr/stampa | Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2020 |
| Descrizione fisica | 1 online resource (342 p.) |
| Soggetto topico |
Biology, life sciences
Research & information: general |
| Soggetto non controllato |
ACE-inhibitory activity
acrylamide airway inflammation alcalase hydrolysate Alzheimer's disease AMD AMP identification and design amyloid amyloid fibrils and endothelial regeneration angiogenic precursor cells angiotensin I converting enzyme anti-biofilm peptides anti-inflammatory antibiotic resistance antifungal activity antigen-specific antihypertensive peptides antimicrobial peptide antimicrobial peptides antimicrobial peptides (AMPs) antimicrobial resistance antioxidant activity antioxidant peptide antiproliferative assay antisepsis, peptide antibiotics apolipoprotein E arthritis asthma Aβ peptide bioactive peptide bioactive peptides biomarkers BIOPEP-UWM database biosynthesis bone erosion cancer antigen cancer stem cells cartilage destruction cathelicidins Cec-analogs Cecropins central nervous system diseases chemoprevention Chlorella sorokiniana chronic diseases Clostridioides difficile CNV collagen collagen peptide colorectal cancer combinatorial library confocal microscopy conjugation copper Crassostrea angulata cryptides CXCR3 cystic fibrosis cytoprotective effect database defensins diseases docetaxel doxorubicin dry-cured pork ham dyslipidemia endothelial dysfunction endothelial progenitor cells energy expenditure enteric nervous system enzyme extra domain B fermentation fetal bovine serum (FBS) fibroblasts fibronectin Fmoc/tBu food intake regulation food-derived foods formyl peptide receptors FPYLRH fresh tissue functional food galanin gender differences glioma GPR10 Histatin-5 host defense peptides Hs02 human antimicrobial peptides human keratinocytes humanized mouse hybrid peptide hydrolysis hydroxyprolyl-glycine (Hyp-Gly) hyperglycemia hypertension immune checkpoint inhibitor immune response immune suppression immunomodulant in silico In situ tetramer staining inflammation inflammatory bowel disease insects intragenic antimicrobial peptide Lactoferricin B (Lfcin B) library design ligands lunasin MDA MDR infectious diseases membrane activity MHC tetramer migration miiuy croaker (Miichthys miiuy) mode of action molecular blind docking molecular docking molecular weight monocyte MRSA multimeric peptides mutagenesis n/a nano liquid chromatography tandem mass spectrometry (nanoLC-nanoESI MS/MS) neuroprotection neurotensin NF-κB non-atopic asthma nutraceuticals nutrition obesity oral delivery osteostatin oxidative stress pegylated glucagon-like peptide 1 peptide peptide vaccine peptide-drug conjugate physico-chemical properties PI3K/Akt pathway pidotimod pig piscidins platelets polymicrobial biofilms pro-inflammatory pro-inflammatory cytokines prolactin-releasing peptide prolyl-hydroxyproline (Pro-Hyp) prostate cancer protection ability proteolysis proteome microarray proteomics pseudin-2 Pseudomonas aeruginosa pulmonary emphysema RF-amide peptides rheumatic diseases screening sheepskin signaling Sjögren's syndrome SMILES code solid-phase synthesis sPLA2 Staphylococcus aureus stomach swim bladder synergistic effects synergy T cell T cells targeting temporin therapeutic potential type 1 diabetes vasoactive intestinal peptide VEGFR1 velvet antler VPAC1 receptor VPAC2 receptor whey peptides Αβ oligomer |
| Formato | Materiale a stampa |
| Livello bibliografico | Monografia |
| Lingua di pubblicazione | eng |
| Altri titoli varianti | Peptides for Health Benefits 2019 |
| Record Nr. | UNINA-9910557492903321 |
Hernández-Ledesma Blanca
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| Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2020 | ||
| Lo trovi qui: Univ. Federico II | ||
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