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Anticancer Agents : Design, Synthesis and Evaluation
Anticancer Agents : Design, Synthesis and Evaluation
Autore Chen Qiao-Hong
Pubbl/distr/stampa Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021
Descrizione fisica 1 online resource (606 p.)
Soggetto topico Medicine and Nursing
Soggetto non controllato 1,2,3-triazole
2H-benzo[e][1,2,4]thiadiazine 1,1-dioxide
3,6-dibromocarbazole
4-(pyridin-4-yloxy)benzamide
5-bromoindole
5-fluorouracil
ABCB1 (P-glycoprotein)
actin
ADME
allene
amides/esters
androgen receptor
anti-cancer activity
anti-neuroinflammation
anti-ovarian cancer
anti-tumor
anticancer
anticancer activity
anticancer agent
anticancer agents
anticancer compounds
antimitotic agents
antioxidant activity
antiproliferative activity
antiproliferative agent
antitumor
antitumor activity
apalutamide
apoptosis
aromatase
benzimidazole
benzofuran-pyrazole
benzofurans
beta-lapachone
bivalency
breast cancer
c-Met
carbazole
cell cycle
chemical synthesis
chemoresistance
chrysin analogues
colchiceine
colchicine amide
colchicine analogs
colchicine sulfonamide
colon cancer
computational docking
coumarin
crystal structure
cyanopyridone
cytotoxic activity
cytotoxic properties
cytotoxicity
darolutamide
DFT study
dihydroartemisinin
dihydropyranoindole
docking
docking studies
drug discovery
drug resistance
E-stereoselective
enzalutamide
enzyme inhibition
estrone derivatives
flavonoid
flavonoids
gemcitabine
HDAC inhibitors
HeLa
HepG2
hydrates
hydrazine
IGF-1R
IL-12
immune modulation
indoleamine 2,3-dioxygenase
inflammation
inhibitor
K562
kinase inhibitor
MCF-7
MDM2-p53 interaction
migration
mimetics
molecular simulation
MOLT-4
multidrug resistance (MDR) reversal
N-substituted pyrazoline
nanoparticles
natural product
neuroblastoma
NIH3T3
o-nitro-benzyl
organosilicon compounds
ortho-quinones
ovarian cancer
overcoming drug resistance
P-glycoprotein
P-MAPA
PARP inhibitor
PARP-1 inhibition
phenylpyrazolopyrimidine
photoactivatable protecting groups
PI3Ks
PI3Kα inhibitor
PI3Kδ inhibitors
polyvalency
prodrug
prostate cancer
PROTACs
protein degradation
protein kinase
protein-protein interactions
Pyrazole
pyrazolopyridine
pyridotriazine
quinazolin-4(3H)-one
quinazolin-4(3H)-thione
regioselective
salinomycin
Schiff base
SILA-409 (Alis-409)
SILA-421 (Alis-421)
Src
substituted pyridine
synergy
synthesis
Talazoparib
tanshione IIA
taxoids
thiazolidinone
Thienopyrimidine
thienopyrimidinone
thiocolchicine
thiopene
thioxotriazopyridine
TLR signaling
topoisomerase II inhibitor
triazolothiadiazine
triple-negative breast cancer
tryptophan metabolism
tubulin inhibitors
tumor specificity
urea
virtual screening
xanthones
yeast-based assays
zampanolide
βIII-tubulin
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Altri titoli varianti Anticancer Agents
Record Nr. UNINA-9910557129103321
Chen Qiao-Hong  
Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021
Materiale a stampa
Lo trovi qui: Univ. Federico II
Opac: Controlla la disponibilità qui
Bioactive Natural Products from the Red Sea
Bioactive Natural Products from the Red Sea
Autore Rateb Mostafa
Pubbl/distr/stampa Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021
Descrizione fisica 1 online resource (152 p.)
Soggetto topico Research & information: general
Soggetto non controllato Actinokineospora
Alternaria
androgen receptor
anti-inflammatory
antibacterial
antibiofilm
antimalarial
antimicrobial
antimicrobial activities
Aspergillus falconensis
azaphilones
bioactivity
biodiversity
ceramide
cerebroside
co-cultivation
co-culture
cytotoxic
cytotoxic activity
diketopiperazine alkaloids
DNA gyrase
docking
docking studies
Epicoccum
epicotripeptin
ergosterol derivative
halogenated 3-phenylpropanoic acid derivatives
LC-HRESIMS
marine actinomycetes
marine metagenomics
marine natural products
marine organisms
metabolic analysis
metabolomics
n/a
neuroprotective
NF-κB inhibition
OSMAC
phenazine
phragamide
pyruvate kinase
Red Sea
Red Sea sponges
Rhodococcus
seagrass
Sinularia polydactyla
soft coral
sponge-associated actinomycetes
steroids
Streptomyces coelicolor LY001
structural determinations
Stylissa carteri
Thalassodendron ciliatum
X-ray diffraction
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Record Nr. UNINA-9910557540903321
Rateb Mostafa  
Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021
Materiale a stampa
Lo trovi qui: Univ. Federico II
Opac: Controlla la disponibilità qui
Cholinesterase Research
Cholinesterase Research
Autore Korabecny Jan
Pubbl/distr/stampa Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021
Descrizione fisica 1 online resource (223 p.)
Soggetto topico Medicine and Nursing
Soggetto non controllato acetylcholinesterase
acetylcholinesterase inhibitor
acetylcholinesterase inhibitors
alkaloids
Alzheimer disease
Alzheimer's disease
Amaryllidaceae
antioxidants
behavior
blood-brain barrier crossing
bone healing
butyrylcholinesterase
butyrylcholinesterase inhibitors
carltonine A-C
catalysis
cholinesterase
dementia
docking
docking studies
donepezil
fluorene
hemostasis
hydrolysis
in silico
in vitro
inhibition
MD simulations
molecular dynamics
molecular modeling
molecular modelling
molecular recognition
multi-target directed ligands
N-methyl-d-aspartate receptor
n/a
Narcissus pseudonarcissus cv. Carlton
neutron scattering
nutraceuticals
organophosphates
organophosphorus
organophosphorus nerve agents
osmotic stress
osseointegration
oxime
pharmacodynamics
phytochemicals
reactivation
reactivation process
reactivators
slow-binding inhibition
transition state analog
ventilation
zebrafish
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Record Nr. UNINA-9910557764703321
Korabecny Jan  
Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021
Materiale a stampa
Lo trovi qui: Univ. Federico II
Opac: Controlla la disponibilità qui