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Anticancer Agents : Design, Synthesis and Evaluation
Anticancer Agents : Design, Synthesis and Evaluation
Autore Chen Qiao-Hong
Pubbl/distr/stampa Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021
Descrizione fisica 1 online resource (606 p.)
Soggetto topico Medicine and Nursing
Soggetto non controllato 1,2,3-triazole
2H-benzo[e][1,2,4]thiadiazine 1,1-dioxide
3,6-dibromocarbazole
4-(pyridin-4-yloxy)benzamide
5-bromoindole
5-fluorouracil
ABCB1 (P-glycoprotein)
actin
ADME
allene
amides/esters
androgen receptor
anti-cancer activity
anti-neuroinflammation
anti-ovarian cancer
anti-tumor
anticancer
anticancer activity
anticancer agent
anticancer agents
anticancer compounds
antimitotic agents
antioxidant activity
antiproliferative activity
antiproliferative agent
antitumor
antitumor activity
apalutamide
apoptosis
aromatase
benzimidazole
benzofuran-pyrazole
benzofurans
beta-lapachone
bivalency
breast cancer
c-Met
carbazole
cell cycle
chemical synthesis
chemoresistance
chrysin analogues
colchiceine
colchicine amide
colchicine analogs
colchicine sulfonamide
colon cancer
computational docking
coumarin
crystal structure
cyanopyridone
cytotoxic activity
cytotoxic properties
cytotoxicity
darolutamide
DFT study
dihydroartemisinin
dihydropyranoindole
docking
docking studies
drug discovery
drug resistance
E-stereoselective
enzalutamide
enzyme inhibition
estrone derivatives
flavonoid
flavonoids
gemcitabine
HDAC inhibitors
HeLa
HepG2
hydrates
hydrazine
IGF-1R
IL-12
immune modulation
indoleamine 2,3-dioxygenase
inflammation
inhibitor
K562
kinase inhibitor
MCF-7
MDM2-p53 interaction
migration
mimetics
molecular simulation
MOLT-4
multidrug resistance (MDR) reversal
N-substituted pyrazoline
nanoparticles
natural product
neuroblastoma
NIH3T3
o-nitro-benzyl
organosilicon compounds
ortho-quinones
ovarian cancer
overcoming drug resistance
P-glycoprotein
P-MAPA
PARP inhibitor
PARP-1 inhibition
phenylpyrazolopyrimidine
photoactivatable protecting groups
PI3Ks
PI3Kα inhibitor
PI3Kδ inhibitors
polyvalency
prodrug
prostate cancer
PROTACs
protein degradation
protein kinase
protein-protein interactions
Pyrazole
pyrazolopyridine
pyridotriazine
quinazolin-4(3H)-one
quinazolin-4(3H)-thione
regioselective
salinomycin
Schiff base
SILA-409 (Alis-409)
SILA-421 (Alis-421)
Src
substituted pyridine
synergy
synthesis
Talazoparib
tanshione IIA
taxoids
thiazolidinone
Thienopyrimidine
thienopyrimidinone
thiocolchicine
thiopene
thioxotriazopyridine
TLR signaling
topoisomerase II inhibitor
triazolothiadiazine
triple-negative breast cancer
tryptophan metabolism
tubulin inhibitors
tumor specificity
urea
virtual screening
xanthones
yeast-based assays
zampanolide
βIII-tubulin
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Altri titoli varianti Anticancer Agents
Record Nr. UNINA-9910557129103321
Chen Qiao-Hong  
Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021
Materiale a stampa
Lo trovi qui: Univ. Federico II
Opac: Controlla la disponibilità qui
Feature Papers in Eng
Feature Papers in Eng
Autore Gil Bravo Antonio
Pubbl/distr/stampa Basel, : MDPI Books, 2022
Descrizione fisica 1 electronic resource (236 p.)
Soggetto topico Technology: general issues
Soggetto non controllato hydrofoil optimization
NSGA-II
CFD
XFOIL
NACA 63815
bezier curve
ultrasound application
glass bottles
fruit juice
foam drainage
foaming behavior
martensitic phase transformation (MPT)
grain misorientation (GMO)
surface roughening (Ra)
grain size (Dg)
solid oxide fuel cell
computational fluid dynamics
sensitivity analysis
optimization
sand retention test
sand control devices
sand production
sand replication
SAGD
probabilistic risk assessment
multi-hazards
nuclear safety
dry-cured ham
food-grade chemical
coating
mechanical performance characteristics
chemical treatment
ham nets
pest management
mechanical test
mesh fabric
artificial magnetic conductor (AMC)
specific absorption rate (SAR)
coplanar waveguide (CPW) antenna
magneto-dielectric (MD)
mobile phones
wireless communications
optical multi-band systems
physical layer modeling
fiber-optic communications
commercially available components
planar transformer
eco-design
environmental impact evaluation
product efficiency
DC-DC converter
dual active bridge (DAB)
life cycle optimization
fuel optimization
low cost HEV
optimum hybridization
bubble nucleation
gas-liquid systems
supersaturation
step-down pressure
Fick's second law diffusion
characteristic time
Q factor
damping model
transitional flow regime
viscous flow regime
MEMS oscillator
bending modes
zirconium phosphate
titanium phosphate
nanolayered phosphates
nanofibrous titanium phosphate
chemical synthesis
crystal structure
technological applications
drug delivery
biomedical applications
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Record Nr. UNINA-9910595068303321
Gil Bravo Antonio  
Basel, : MDPI Books, 2022
Materiale a stampa
Lo trovi qui: Univ. Federico II
Opac: Controlla la disponibilità qui
Magnetic Nanomaterials
Magnetic Nanomaterials
Autore Del Bianco Lucia
Pubbl/distr/stampa Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022
Descrizione fisica 1 online resource (234 p.)
Soggetto topico History of engineering & technology
Technology: general issues
Soggetto non controllato bone tissue engineering
Burstein-Moss shift
cell labelling
chemical synthesis
CoFeB
core/shell nanoparticles
density functional theory
disordered magnetism
electrodeposition technique
epitaxial Ni-Mn-Ga films
exchange bias
Fe-oxide nanocrystallites
FePd alloy
ferrimagnetic materials
glassy correlation length
Heusler alloys
hybrid systems
III-nitrides
interlayer exchange coupling
iron nitrides
Kubelka-Munk function
magnetic aggregates
magnetic anisotropy
magnetic freezing
magnetic heating
magnetic hyperthermia
magnetic hysteresis
magnetic interactions
magnetic materials
magnetic nanoparticles
magnetic properties
magnetic shape memory alloys
magneto-sonoporation
magnetron sputtering
martensitic transition
mixed nanoparticle systems
multicore nanoparticles
nanocomposites
nanocrystals
nanogranular Au/Fe-oxide
nanoparticles
nanowires
osteogenesis
Raman spectroscopy
sol-gel
stem cells
structural characterisation
substitutional doping
super-spin glass
superparamagnetic iron oxide particles
superparamagnetism
synthetic antiferromagnet
thermally assisted magnetic scanning probe lithography
transmission electron microscopy
twin boundary
ultrasounds
UV-blue photoluminescence
vibrating sample magnetometry
ZnNiO
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Record Nr. UNINA-9910557610803321
Del Bianco Lucia  
Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022
Materiale a stampa
Lo trovi qui: Univ. Federico II
Opac: Controlla la disponibilità qui
Marine Bioactive Peptides : : Structure, Function, and Therapeutic Potential / / Tatiana V. Ovchinnikova
Marine Bioactive Peptides : : Structure, Function, and Therapeutic Potential / / Tatiana V. Ovchinnikova
Autore Ovchinnikova Tatiana V
Pubbl/distr/stampa MDPI - Multidisciplinary Digital Publishing Institute, 2019
Descrizione fisica 1 electronic resource (442 p.)
Soggetto topico Biology, life sciences
Soggetto non controllato cone snail
tilapia
animal models
BRICHOS domain
recombinant peptide
calcium absorption
plastein reaction
antioxidant activity
endothelial dysfunction
C3a
lung cancer
invertebrate immunity
identification
zinc bioavailability
NA-inhibitory peptide
nuclear magnetic resonance (NMR)
review
ACE-inhibitory activity
intestinal absorption
hairtail (Trichiurus japonicas)
DU-145 cells
peptide
crustacean
venom duct
Kalloconus
drug design
molecular symmetry
arenicin
?-helix
APETx2
conotoxins
functional diversity
docking
conotoxin
neuraminidase
angiotensin II
polychaeta
influenza virus
phylogeny
gene expression
host defense peptide
Perinereis aibuhitensis
anti-diabetic activity
conopeptides
SHRs
Chlorella pyrenoidosa protein hydrolysate (CPPH)
metastasis
Caco-2 cell monolayer
Nrf2
caco-2 cells
HUVEC
PYP15
sea cucumber
decapeptide
cytotoxic
arenicin-1
marine peptides
cell proliferation
Conus
Conus ateralbus
self-production of hydrogen peroxide
antimicrobial activity
molecular dynamics
machine learning
tachyplesins
ion channels
gut microbiota
Anthopleura anjunae oligopeptide
signaling pathways
half-fin anchovy hydrolysates
NF-?B
Chlorella pyrenoidosa protein hydrolysate-calcium chelate (CPPH-Ca)
antihypertensive effect
QAGLSPVR
antimicrobial peptides
vasculogenic mimicry
antibacterial
?-hairpin
innate immunity
transcriptome sequencing
HIF-1?
Gracilariopsis lemaneiformis
function
ACE-inhibitory peptide
complement
peptide-zinc complex
structure-activity relationship
multi-functional peptides
cod skin
adsorption
Maillard reaction products
molecular docking
antibacterial peptide
PI3K/AKT/mTOR signaling pathway
Arenicola marina
antimicrobial peptide
Rana-box
acid-sensing ion channel
Neptunea arthritica cumingii
apoptosis
membrane damage
proteolytic system
toxin
polyphemusins
computational studies
muscle
oyster zinc-binding peptide
abalone
pain relief
transport routes
cytotoxicity
dexamethasone
cell death
host?microbe relationship
anti-LPS factor
MMPs
protein synthesis
structure
Pyropia yezoensis peptide
cone snails
chemical synthesis
prostate cancer
Ugr 9-1
myotube atrophy
ISBN 9783039215331
3039215337
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Record Nr. UNINA-9910367750603321
Ovchinnikova Tatiana V  
MDPI - Multidisciplinary Digital Publishing Institute, 2019
Materiale a stampa
Lo trovi qui: Univ. Federico II
Opac: Controlla la disponibilità qui
Strategies to Improve Antineoplastic Activity of Drugs in Cancer Progression
Strategies to Improve Antineoplastic Activity of Drugs in Cancer Progression
Autore Stefanachi Angela
Pubbl/distr/stampa Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022
Descrizione fisica 1 electronic resource (416 p.)
Soggetto topico Research & information: general
Biology, life sciences
Soggetto non controllato EGR-1
flavonoid
(E)-5-((4-oxo-4H-chromen-3-yl)methyleneamino)-1-phenyl-1H-pyrazole-4-carbonitrile
MDA-MB-231
MMP9
TNFα
pancreatic ductal adenocarcinoma
cyclodextrin inclusion complex
phase solubility studies
preformulation studies
biphenylnicotinamide derivatives
dual inhibitor
EGFR
VEGFR2
ligand-based pharmacophore
molecular docking
molecular dynamics
leukemias
doxorubicin
inflammation
drug delivery
tumor targeting
elastin-like polypeptide
cell penetrating peptide
matrix metalloproteinase
doxorubicin resistance
photosensitizer delivery system
PAMAM dendrimer
photodynamic therapy
cytotoxicity
phototoxicity
colorectal adenocarcinoma
dicarboximides
chemical synthesis
apoptosis
kinases
anticancer
gene profiling
SAR
biomarkers
colorectal cancer
early detection examination
liquid biopsy
personalized medicine
tumor treatment
exosomes
ctDNA
CTC
cytotoxic activity
pyrazole derivatives
MTT assay
ADMET analysis
single-crystal diffraction
FTIR spectroscopy
NMR spectroscopy thermogravimetric analysis
acute myelogenous leukemia
platelets
microparticles
γδ T cells
immunotherapy
tumor resistance
combination therapy
tumor microenvironment
immune checkpoint inhibitor
neuroblastoma
molecular iodine
cyclophosphamide
xenografts
metronomic therapy
tamoxifen
CYP2D6
MCF-7
Ishikawa cells
SERM
TNBC
uterotrophic
α-mangostin
poly(amidoamine) dendrimer
targeted drug delivery
biotin targeting
glioblastoma multiforme
squamous cell carcinoma
antiparasitic therapy
diclofenac
indomethacin
oleanolic acid derivative conjugates
NF-κB
Nrf2
MAPKs
PSN-1 cells
reactive oxygen species
glioblastoma
brain tumor
extracellular vesicles
pancreatic cancer
paclitaxel
clathrin
endocytosis
sulforaphane
nicotine
metalloproteinase-9
gastric cancer
cell invasion
Arylquin 1
colon cancer
tumor progression
azelastine
oxidative stress
autophagy
mitotic catastrophe
chronic myeloid leukemia
imatinib
tyrosine kinase
ketoconazole
P-glycoprotein
drug efflux transporter
non-small-cell lung cancer
cisplatin resistance
aldehyde dehydrogenase
isothiocyanates
disulfiram
epithelial to mesenchymal transition
aminopeptidase N
acetamidophenones
Schiff bases
semicarbazones
thiosemicarbazones
inhibition of proliferation
ISBN 3-0365-5927-2
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Record Nr. UNINA-9910639990003321
Stefanachi Angela  
Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022
Materiale a stampa
Lo trovi qui: Univ. Federico II
Opac: Controlla la disponibilità qui
Sulfur-Containing Marine Bioactives
Sulfur-Containing Marine Bioactives
Autore Palumbo Anna
Pubbl/distr/stampa Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021
Descrizione fisica 1 online resource (140 p.)
Soggetto topico Medicine
Soggetto non controllato adjuvant
age-related macular degeneration
aggregates
algae
angiogenesis
anti-settlement
antioxidant
antioxidant capacity
autotrophic culture
biofouling
brown seaweed extracts
carbohydrate sulfotransferase
carrageenan
chemical synthesis
colloid
cytochrome P450
cytotoxic effects on tumor cells
diatoms
eco-friendly
exopolysaccharides
FGF2
fucan
fucoidan
galactose-6 sulfurylase
gallic acid
heterotrophic culture
immunomodulatory activity
invasion
Laminaria hyperborea
light
marine coatings
MMP-2
MMP-9
molecular weight
natural products
nitric oxide
ovothiol
oxidative stress
proliferation
propylene glycol alginate sodium sulfate
rare actinobacteria
red alga
reproduction stages
retinal pigment epithelium
screening
structure elucidation
sulfated
sulfavants
Tetraselmis suecica
thiopeptide antibiotic
VEGF
WD 40
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Record Nr. UNINA-9910557113603321
Palumbo Anna  
Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021
Materiale a stampa
Lo trovi qui: Univ. Federico II
Opac: Controlla la disponibilità qui
Synthesis of Marine Natural Products and Molecules Inspired by Marine Substances II
Synthesis of Marine Natural Products and Molecules Inspired by Marine Substances II
Autore Manzo Emiliano
Pubbl/distr/stampa Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021
Descrizione fisica 1 online resource (111 p.)
Soggetto topico Chemistry
Research & information: general
Soggetto non controllato (−)-majusculoic acid
ADMET
animal studies
anti-inflammation
aureol
Avicennia alba
biological activity
biosynthesis
cancer
cardiovascular diseases
CCK-8
chemical synthesis
cyclomarins
cyclopeptides
divergent total synthesis
gag polyprotein
homology modeling
ilamycins
In-silico drug design
inflammation
LPS
malaria
marine alkaloids
marine natural products
molecular dynamics simulation
n/a
natural products
rufomycins
tetracyclic meroterpenoids
total synthesis
tuberculosis
virtual screening
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Record Nr. UNINA-9910557724503321
Manzo Emiliano  
Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021
Materiale a stampa
Lo trovi qui: Univ. Federico II
Opac: Controlla la disponibilità qui