Anticancer Inhibitors
| Anticancer Inhibitors |
| Autore | Fantacuzzi Marialuigia |
| Pubbl/distr/stampa | Basel, : MDPI Books, 2022 |
| Descrizione fisica | 1 electronic resource (216 p.) |
| Soggetto topico |
Research & information: general
Chemistry |
| Soggetto non controllato |
breast cancer
tamoxifen LY294002 synergism apoptosis cell cycle tea (Camellia sinensis) flowers BTFS A2780/CP70 ovarian cancer cells S phase cell cycle arrest nicotinamide phosphoribosyltransferase NAD+ biosynthesis inhibitor azacyclohexane anticancer drug drug design enthalpy effect NSCLC Cathepsin K cell proliferation cell migration cell invasion mTOR isatin-hydrazones cytotoxicity CDK2 inhibitor ATP competitive inhibitor ADME analysis receptor tyrosine kinases protein-protein interactions protein engineering directed evolution angiogenesis binding affinity agonistic activity saponins phytochemicals tea (Camellia sinensis) flower ovarian cancer autophagy ZMYND8 tumorigenesis epigenetic regulation pro-oncogenic effects tumor suppression tacrine-coumarin derivatives DNA topoisomerases I, II lung carcinoma cells A549 chemotherapy prodrug drug targeting overexpressed enzymes ADC ADEPT GDEPT LEAPT PROTAC cyclin-dependent kinase cancer resistance small molecule inhibitors PROTACs statins pancreatic cancer DNA microarray pitavastatin cerivastatin simvastatin fluvastatin atorvastatin pravastatin HMG-CoA reductase inhibitors |
| Formato | Materiale a stampa |
| Livello bibliografico | Monografia |
| Lingua di pubblicazione | eng |
| Record Nr. | UNINA-9910595069203321 |
Fantacuzzi Marialuigia
|
||
| Basel, : MDPI Books, 2022 | ||
| Lo trovi qui: Univ. Federico II | ||
| ||
Novel Anti-cancer Agents and Cellular Targets and Their Mechanism(s) of Action
| Novel Anti-cancer Agents and Cellular Targets and Their Mechanism(s) of Action |
| Autore | Allison Simon J |
| Pubbl/distr/stampa | MDPI - Multidisciplinary Digital Publishing Institute, 2022 |
| Descrizione fisica | 1 online resource (206 p.) |
| Soggetto topico |
History of engineering & technology
Technology: general issues |
| Soggetto non controllato |
5-FU resistance
8-hydroxydaidzein affibody drug conjugate (AffiDC) affibody molecule albumin binding domain angiogenesis anti-cancer agent anticancer drug apoptosis AQ4N autophagy B-lactam steroid alkylators BCR-ABL biomarker bioprecursor breast cancer BxPC-3 c-myc cancer hallmarks CCN1 colorectal cancer Connectivity Map CYP1A1 CYP1B1 CYP2W1 Cytochrome P450 DM1 drug repurposing duocarmycin EGFR tyrosine kinase inhibitor emtansine expression gene silencing Genomics of Drug Sensitivity in Cancer glioblastoma HepG2 Huh7 human epidermal growth factor receptor 3 (HER3) hybrid steroidal alkylating agents in vivo imaging invasion isatin sulfonamides K562 MAPK mesenchymal-amoeboid transition microtubule acetylation migration molecular docking n/a nanoparticles nanosystems NF-κB oncogene ovarian cancer phortress photon upconversion PLGA poly (ADP-ribose) polymerase inhibitors prodrug RNA interference siRNA synthetic lethality triple-negative breast cancer triplet-triplet annihilation |
| ISBN | 3-0365-5222-7 |
| Formato | Materiale a stampa |
| Livello bibliografico | Monografia |
| Lingua di pubblicazione | eng |
| Altri titoli varianti | Novel Anti-cancer Agents and Cellular Targets and Their Mechanism |
| Record Nr. | UNINA-9910619465503321 |
Allison Simon J
|
||
| MDPI - Multidisciplinary Digital Publishing Institute, 2022 | ||
| Lo trovi qui: Univ. Federico II | ||
| ||
Novel Strategies in the Development of New Therapies, Drug Substances and Drug Carriers
| Novel Strategies in the Development of New Therapies, Drug Substances and Drug Carriers |
| Autore | Kutner Andrzej |
| Pubbl/distr/stampa | Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022 |
| Descrizione fisica | 1 online resource (450 p.) |
| Soggetto topico |
Chemistry
Research & information: general |
| Soggetto non controllato |
1,2,4-triazole
25 vitamin D 24-hydroxylase A-ring active substance delivery systems active substance-controlled release ADME alkaloids alpha-ketoglutarate analogue actions at genes anti-depressant therapy anti-inflammatory activity anticancer activity anticancer drug anticancer drugs antidepressants antimalarial antimicrobial activity antimicrobial compounds antimicrobial peptide (AMP) antioxidant activity antiparasitic agents antiviral proteins apoptosis Au(III) complex biomarker biomedical hydrogels calcilytic calcimimetic calcium-sensing receptor cancer cancer cells cancer therapy cancer treatment CD-ring cell cycle cell invasion cell migration Chelidonium majus ChIP-chip analysis colon cancer colorectal cancer copper (II) complexes CRISPR/Cas9 cyclooxygenase CYP24A1 CYP24A1-dependent metabolism CYP27B1 cytotoxic activity cytotoxic study cytotoxicity defense-related proteins depression dermaseptin distal enhancers drug drug design drug design and discovery drug discovery dual 5-HT1A/SERT activity electrochemistry enantiomer fluorine frog skin peptides genistein genome editing glucose metabolism glycoconjugates gold gold electrode greater celandine hemolysis high-grade serous ovarian cancer cells histone deacetylase (HDAC) histone H3 acetylation HT-29 human DNA topoisomerase hydrogels for cosmetology hydrogels for dermatology IL-8 inflammation JNK latex LHRH lung cancer major latex protein MALDI metabolite metallodrugs methotrexate molecular docking molecular modeling multimodal activity n/a nanoparticles organometallic oxidation mechanisms Phyllomedusa bicolor Plasmodium falciparum (P. falciparum) PRI-2191 proliferation prostate cancer proteome analysis pyridazinone pyrido[1,2-c]pyrimidines resveratrol rickets RNA polymerase II SAR self-assembled monolayer side-chain spectroscopic data split luciferase-based biosensor stereospecificity synthesis targeted therapy tetrahydro-β-carbolines TGF-β therapeutic peptides thiourea transcription transdermal active substance delivery systems VEGF vitamin D vitamin D analogs vitamin D biology and action vitamin D hormone (1,25(OH)2D3) vitamin D receptor vitamin D3 Warburg effect |
| Formato | Materiale a stampa |
| Livello bibliografico | Monografia |
| Lingua di pubblicazione | eng |
| Record Nr. | UNINA-9910585938903321 |
Kutner Andrzej
|
||
| Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022 | ||
| Lo trovi qui: Univ. Federico II | ||
| ||
Nucleic Acids Conjugates for Biotechnological Applications
| Nucleic Acids Conjugates for Biotechnological Applications |
| Autore | Endoh Tamaki |
| Pubbl/distr/stampa | Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021 |
| Descrizione fisica | 1 online resource (130 p.) |
| Soggetto topico | Technology: general issues |
| Soggetto non controllato |
abasic site
anticancer drug aptamer artificial viral capsid BRET-based biosensor camptothecin derivative catalytic RNA cellular uptake conjugate crosslink cytosine methyltransferase cytotoxicity DNA DNA aptamer DNA-protein conjugate drug delivery drug delivery system encapsulation fluorescent probe fluorescent sensors group I ribozyme invasion irinotecan macrophages microRNA mRNA multiple sclerosis n/a nanocapsule nanoparticles NLS nucleic acid binding protein oligonucleotide peptide-DNA conjugate PNA poly(A) tail PUF replication initiation protein repulsive guidance molecule a ribonucleopeptide (RNP) RNA binding protein RNA nanostructure RNA nanotechnology RNA regulation RNA-peptide conjugate RNA-protein complex Schiff base self-assembly small interfering RNA therapeutic nucleic acid trans-splicing β-annulus peptide |
| Formato | Materiale a stampa |
| Livello bibliografico | Monografia |
| Lingua di pubblicazione | eng |
| Record Nr. | UNINA-9910669804103321 |
Endoh Tamaki
|
||
| Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021 | ||
| Lo trovi qui: Univ. Federico II | ||
| ||
Role of Natural Bioactive Compounds in the Rise and Fall of Cancers : Volume 2
| Role of Natural Bioactive Compounds in the Rise and Fall of Cancers : Volume 2 |
| Autore | Luparello Claudio |
| Pubbl/distr/stampa | Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2020 |
| Descrizione fisica | 1 online resource (318 p.) |
| Soggetto topico |
Biology, life sciences
Research and information: general |
| Soggetto non controllato |
acute myeloid leukemia
adipocyte inflammation AKT AMPK angiogenesis anti-cancer drug anti-proliferative anticancer anticancer activities anticancer drug anticancer drugs AOM/DSS model apoptosis autophagy berberine Berthel bioactivities bioavailability brain cancer breast cancer breast cancer cells breast cancer prognostic breast cancer risk Calocedrus formosana cancer cancer metabolism cancer stem cell cancer therapy carrageenan caspase-independent cell death cell death cell signaling cell-cycle arrest chemoprevention colchicine alkaloid colon cancer colon cancer cells colorectal cancer daidzein daidzein metabolites drugs EGCG EGFR signaling EGFR TKI eicosapentaenoic acid epigallocatechin-3-gallate (EGCG) epithelial mesenchymal transition ER stress estrogen estrogen receptor alpha ethanol experimental therapeutics FASN inhibitors flavonoids formononetin fucoidan G2/M arrest gallic acid gemcitabine gigantol gliomas glucose transport glycolysis glycolytic markers HDAC HO-1 honokiol human cancer cells immunotherapy inflammation innate immunity invasion isobolography isorhamnetin JAK/STAT lung cancer malignant cancer malignant tumors of the peripheral nerve sheath (MPNST) Malva pseudolavatera Webb & mangrove marine sponge mechanism melanoma cells mesoporous silica nanoparticles metastasis microRNAs MMPs molecular mechanisms multiple myeloma n/a nanoparticle-based delivery systems natural anti-inflammatory compounds natural bioactive compound natural compounds natural polyphenols natural product neurofibromas nicotine nobiletin non-coding RNAs Nrf2 NSCLC nutrition obesity oleacein oleuropein olive leaf extract oncogenic cascades oral cancer inhibition p53 paclitaxel pancreatic cancer PD-1 immune checkpoint inhibitor and cancer immunotherapy PD-L1 persistent organic pollutants phosphofructokinase phytochemicals Piper eriopodon, alkenylphenols polyphenols preclinical models pro-resolving lipids proteomics RacGAP1 radiotherapy reactive oxygen species renin-angiotensin system resistance ROS schwannomas Seahorse analysis signaling pathways signalling pathway small organic agents STAT3 Streptomyces systematic review targeted delivery system TRAIL tumor density tumor maintenance uterine sarcoma xenograft Xenopus laevis XIAP antagonists XIAP-BIR3 domain yatein α9-nAChR β-glucans |
| Formato | Materiale a stampa |
| Livello bibliografico | Monografia |
| Lingua di pubblicazione | eng |
| Altri titoli varianti | Role of Natural Bioactive Compounds in the Rise and Fall of Cancers |
| Record Nr. | UNINA-9910557476303321 |
Luparello Claudio
|
||
| Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2020 | ||
| Lo trovi qui: Univ. Federico II | ||
| ||
Synthesis, Study and Utilization of Natural Products
| Synthesis, Study and Utilization of Natural Products |
| Autore | Drasar Pavel B |
| Pubbl/distr/stampa | MDPI - Multidisciplinary Digital Publishing Institute, 2020 |
| Descrizione fisica | 1 online resource (234 p.) |
| Soggetto topico | Technology: general issues |
| Soggetto non controllato |
4-epi-varioxiranol A
absolute structure adhesive anti-inflammation anticancer drug antioxidant antioxidant activity apo-CpcB apoptosis bardoxolone methyl bioactivity biosynthesis bromelain caffeoylquinic acids cancer cells cell opening chlorogenic acid cytotoxicity derivatives Emericella variecolor fatty acid flavonoids flexible polyurethane foam flow cytometry gene expression genetical transformation ginkgolide HepG2 cells inhibitor insect sex pheromone isosorbide lipid-lowering effects live-cell fluorescence microscopy melatonin microbial biosynthesis mitochondria n/a natural enantiomer natural product natural products octadecanoid oleic acid-elicited PEGylated purpurin 18 pharmacokinetic features pharmacological activities phenolic acid photodynamic therapy photosensitizer phototoxicity phycocyanin pinocembrin Plantago depressa platelet-activating factor receptor polyphenol polysaccharides post-translationally modified peptides radical scavenger Ramulus mori research progress resource chemistry reversible urethane linkages rheumatoid arthritis ribosomally synthesized RiPP salt stress singlet oxygen SlCOMT1 soy protein isolate Spirulina stilbene synthesis of natural products tea tussock moth tomato total synthesis triglycidylamine triterpenoids varioxiranol A viscosity water resistance |
| ISBN | 3-03928-153-4 |
| Formato | Materiale a stampa |
| Livello bibliografico | Monografia |
| Lingua di pubblicazione | eng |
| Record Nr. | UNINA-9910372783503321 |
Drasar Pavel B
|
||
| MDPI - Multidisciplinary Digital Publishing Institute, 2020 | ||
| Lo trovi qui: Univ. Federico II | ||
| ||
Unconventional Anticancer Metallodrugs and Strategies to Improve their Pharmacological Profile / Maria Contel
| Unconventional Anticancer Metallodrugs and Strategies to Improve their Pharmacological Profile / Maria Contel |
| Autore | Contel Maria |
| Pubbl/distr/stampa | MDPI - Multidisciplinary Digital Publishing Institute, 2019 |
| Descrizione fisica | 1 electronic resource (204 p.) |
| Soggetto topico | Biology, life sciences |
| Soggetto non controllato |
?-? stacking
encapsulation oxindolimine-metal complexes cyclodextrin platinum iodido complexes distribution coefficient antiproliferative activity anticancer agents nanotubes ruthenium platinum Log kw nanoparticles drug discovery metal complex metallodrugs isatin-derived ligands anticancer drug upconverting nanoparticles pyridine benzimidazole dendrimers liposomes thiophene angiogenesis micelles HSA oxidation platinum(IV) imaging chromatographic lipophilicity parameter amidophosphine copper and iron chelators in cancer Log P biomacromolecules bones DNA cleavage stopped-flow spectroscopy silver phosphonates transmetalation metallomics MRI fluorescence quenching partition coefficient gold fingers anticancer HSA binding gold ?0 targeting metastasis DNA interaction antimigration cytotoxicity HPLC ruthenium complexes zinc finger proteins Gold(III) complexes aquaporins antiproliferative protein-DNA recognition photoactivation lipophilicity cancer 1-methylcytosine PET |
| ISBN |
9783039213160
3039213164 |
| Formato | Materiale a stampa |
| Livello bibliografico | Monografia |
| Lingua di pubblicazione | eng |
| Record Nr. | UNINA-9910367755103321 |
Contel Maria
|
||
| MDPI - Multidisciplinary Digital Publishing Institute, 2019 | ||
| Lo trovi qui: Univ. Federico II | ||
| ||