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Anticancer Inhibitors
Anticancer Inhibitors
Autore Fantacuzzi Marialuigia
Pubbl/distr/stampa Basel, : MDPI Books, 2022
Descrizione fisica 1 electronic resource (216 p.)
Soggetto topico Research & information: general
Chemistry
Soggetto non controllato breast cancer
tamoxifen
LY294002
synergism
apoptosis
cell cycle
tea (Camellia sinensis) flowers
BTFS
A2780/CP70 ovarian cancer cells
S phase cell cycle arrest
nicotinamide phosphoribosyltransferase
NAD+ biosynthesis
inhibitor
azacyclohexane
anticancer drug
drug design
enthalpy effect
NSCLC
Cathepsin K
cell proliferation
cell migration
cell invasion
mTOR
isatin-hydrazones
cytotoxicity
CDK2 inhibitor
ATP competitive inhibitor
ADME analysis
receptor tyrosine kinases
protein-protein interactions
protein engineering
directed evolution
angiogenesis
binding affinity
agonistic activity
saponins
phytochemicals
tea (Camellia sinensis) flower
ovarian cancer
autophagy
ZMYND8
tumorigenesis
epigenetic regulation
pro-oncogenic effects
tumor suppression
tacrine-coumarin derivatives
DNA
topoisomerases I, II
lung carcinoma cells
A549
chemotherapy
prodrug
drug targeting
overexpressed enzymes
ADC
ADEPT
GDEPT
LEAPT
PROTAC
cyclin-dependent kinase
cancer
resistance
small molecule inhibitors
PROTACs
statins
pancreatic cancer
DNA microarray
pitavastatin
cerivastatin
simvastatin
fluvastatin
atorvastatin
pravastatin
HMG-CoA reductase inhibitors
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Record Nr. UNINA-9910595069203321
Fantacuzzi Marialuigia  
Basel, : MDPI Books, 2022
Materiale a stampa
Lo trovi qui: Univ. Federico II
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Novel Anti-cancer Agents and Cellular Targets and Their Mechanism(s) of Action
Novel Anti-cancer Agents and Cellular Targets and Their Mechanism(s) of Action
Autore Allison Simon J
Pubbl/distr/stampa MDPI - Multidisciplinary Digital Publishing Institute, 2022
Descrizione fisica 1 online resource (206 p.)
Soggetto topico History of engineering & technology
Technology: general issues
Soggetto non controllato 5-FU resistance
8-hydroxydaidzein
affibody drug conjugate (AffiDC)
affibody molecule
albumin binding domain
angiogenesis
anti-cancer agent
anticancer drug
apoptosis
AQ4N
autophagy
B-lactam steroid alkylators
BCR-ABL
biomarker
bioprecursor
breast cancer
BxPC-3
c-myc
cancer hallmarks
CCN1
colorectal cancer
Connectivity Map
CYP1A1
CYP1B1
CYP2W1
Cytochrome P450
DM1
drug repurposing
duocarmycin
EGFR tyrosine kinase inhibitor
emtansine
expression
gene silencing
Genomics of Drug Sensitivity in Cancer
glioblastoma
HepG2
Huh7
human epidermal growth factor receptor 3 (HER3)
hybrid steroidal alkylating agents
in vivo imaging
invasion
isatin sulfonamides
K562
MAPK
mesenchymal-amoeboid transition
microtubule acetylation
migration
molecular docking
n/a
nanoparticles
nanosystems
NF-κB
oncogene
ovarian cancer
phortress
photon upconversion
PLGA
poly (ADP-ribose) polymerase inhibitors
prodrug
RNA interference
siRNA
synthetic lethality
triple-negative breast cancer
triplet-triplet annihilation
ISBN 3-0365-5222-7
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Altri titoli varianti Novel Anti-cancer Agents and Cellular Targets and Their Mechanism
Record Nr. UNINA-9910619465503321
Allison Simon J  
MDPI - Multidisciplinary Digital Publishing Institute, 2022
Materiale a stampa
Lo trovi qui: Univ. Federico II
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Novel Strategies in the Development of New Therapies, Drug Substances and Drug Carriers
Novel Strategies in the Development of New Therapies, Drug Substances and Drug Carriers
Autore Kutner Andrzej
Pubbl/distr/stampa Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022
Descrizione fisica 1 online resource (450 p.)
Soggetto topico Chemistry
Research & information: general
Soggetto non controllato 1,2,4-triazole
25 vitamin D 24-hydroxylase
A-ring
active substance delivery systems
active substance-controlled release
ADME
alkaloids
alpha-ketoglutarate
analogue actions at genes
anti-depressant therapy
anti-inflammatory activity
anticancer activity
anticancer drug
anticancer drugs
antidepressants
antimalarial
antimicrobial activity
antimicrobial compounds
antimicrobial peptide (AMP)
antioxidant activity
antiparasitic agents
antiviral proteins
apoptosis
Au(III) complex
biomarker
biomedical hydrogels
calcilytic
calcimimetic
calcium-sensing receptor
cancer
cancer cells
cancer therapy
cancer treatment
CD-ring
cell cycle
cell invasion
cell migration
Chelidonium majus
ChIP-chip analysis
colon cancer
colorectal cancer
copper (II) complexes
CRISPR/Cas9
cyclooxygenase
CYP24A1
CYP24A1-dependent metabolism
CYP27B1
cytotoxic activity
cytotoxic study
cytotoxicity
defense-related proteins
depression
dermaseptin
distal enhancers
drug
drug design
drug design and discovery
drug discovery
dual 5-HT1A/SERT activity
electrochemistry
enantiomer
fluorine
frog skin peptides
genistein
genome editing
glucose metabolism
glycoconjugates
gold
gold electrode
greater celandine
hemolysis
high-grade serous ovarian cancer cells
histone deacetylase (HDAC)
histone H3 acetylation
HT-29
human DNA topoisomerase
hydrogels for cosmetology
hydrogels for dermatology
IL-8
inflammation
JNK
latex
LHRH
lung cancer
major latex protein
MALDI
metabolite
metallodrugs
methotrexate
molecular docking
molecular modeling
multimodal activity
n/a
nanoparticles
organometallic
oxidation mechanisms
Phyllomedusa bicolor
Plasmodium falciparum (P. falciparum)
PRI-2191
proliferation
prostate cancer
proteome analysis
pyridazinone
pyrido[1,2-c]pyrimidines
resveratrol
rickets
RNA polymerase II
SAR
self-assembled monolayer
side-chain
spectroscopic data
split luciferase-based biosensor
stereospecificity
synthesis
targeted therapy
tetrahydro-β-carbolines
TGF-β
therapeutic peptides
thiourea
transcription
transdermal active substance delivery systems
VEGF
vitamin D
vitamin D analogs
vitamin D biology and action
vitamin D hormone (1,25(OH)2D3)
vitamin D receptor
vitamin D3
Warburg effect
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Record Nr. UNINA-9910585938903321
Kutner Andrzej  
Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022
Materiale a stampa
Lo trovi qui: Univ. Federico II
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Nucleic Acids Conjugates for Biotechnological Applications
Nucleic Acids Conjugates for Biotechnological Applications
Autore Endoh Tamaki
Pubbl/distr/stampa Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021
Descrizione fisica 1 online resource (130 p.)
Soggetto topico Technology: general issues
Soggetto non controllato abasic site
anticancer drug
aptamer
artificial viral capsid
BRET-based biosensor
camptothecin derivative
catalytic RNA
cellular uptake
conjugate
crosslink
cytosine methyltransferase
cytotoxicity
DNA
DNA aptamer
DNA-protein conjugate
drug delivery
drug delivery system
encapsulation
fluorescent probe
fluorescent sensors
group I ribozyme
invasion
irinotecan
macrophages
microRNA
mRNA
multiple sclerosis
n/a
nanocapsule
nanoparticles
NLS
nucleic acid binding protein
oligonucleotide
peptide-DNA conjugate
PNA
poly(A) tail
PUF
replication initiation protein
repulsive guidance molecule a
ribonucleopeptide (RNP)
RNA binding protein
RNA nanostructure
RNA nanotechnology
RNA regulation
RNA-peptide conjugate
RNA-protein complex
Schiff base
self-assembly
small interfering RNA
therapeutic nucleic acid
trans-splicing
β-annulus peptide
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Record Nr. UNINA-9910669804103321
Endoh Tamaki  
Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021
Materiale a stampa
Lo trovi qui: Univ. Federico II
Opac: Controlla la disponibilità qui
Role of Natural Bioactive Compounds in the Rise and Fall of Cancers : Volume 2
Role of Natural Bioactive Compounds in the Rise and Fall of Cancers : Volume 2
Autore Luparello Claudio
Pubbl/distr/stampa Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2020
Descrizione fisica 1 online resource (318 p.)
Soggetto topico Biology, life sciences
Research and information: general
Soggetto non controllato acute myeloid leukemia
adipocyte inflammation
AKT
AMPK
angiogenesis
anti-cancer drug
anti-proliferative
anticancer
anticancer activities
anticancer drug
anticancer drugs
AOM/DSS model
apoptosis
autophagy
berberine
Berthel
bioactivities
bioavailability
brain cancer
breast cancer
breast cancer cells
breast cancer prognostic
breast cancer risk
Calocedrus formosana
cancer
cancer metabolism
cancer stem cell
cancer therapy
carrageenan
caspase-independent cell death
cell death
cell signaling
cell-cycle arrest
chemoprevention
colchicine alkaloid
colon cancer
colon cancer cells
colorectal cancer
daidzein
daidzein metabolites
drugs
EGCG
EGFR signaling
EGFR TKI
eicosapentaenoic acid
epigallocatechin-3-gallate (EGCG)
epithelial mesenchymal transition
ER stress
estrogen
estrogen receptor alpha
ethanol
experimental therapeutics
FASN inhibitors
flavonoids
formononetin
fucoidan
G2/M arrest
gallic acid
gemcitabine
gigantol
gliomas
glucose transport
glycolysis
glycolytic markers
HDAC
HO-1
honokiol
human cancer cells
immunotherapy
inflammation
innate immunity
invasion
isobolography
isorhamnetin
JAK/STAT
lung cancer
malignant cancer
malignant tumors of the peripheral nerve sheath (MPNST)
Malva pseudolavatera Webb &
mangrove
marine sponge
mechanism
melanoma cells
mesoporous silica nanoparticles
metastasis
microRNAs
MMPs
molecular mechanisms
multiple myeloma
n/a
nanoparticle-based delivery systems
natural anti-inflammatory compounds
natural bioactive compound
natural compounds
natural polyphenols
natural product
neurofibromas
nicotine
nobiletin
non-coding RNAs
Nrf2
NSCLC
nutrition
obesity
oleacein
oleuropein
olive leaf extract
oncogenic cascades
oral cancer inhibition
p53
paclitaxel
pancreatic cancer
PD-1 immune checkpoint inhibitor and cancer immunotherapy
PD-L1
persistent organic pollutants
phosphofructokinase
phytochemicals
Piper eriopodon, alkenylphenols
polyphenols
preclinical models
pro-resolving lipids
proteomics
RacGAP1
radiotherapy
reactive oxygen species
renin-angiotensin system
resistance
ROS
schwannomas
Seahorse analysis
signaling pathways
signalling pathway
small organic agents
STAT3
Streptomyces
systematic review
targeted delivery system
TRAIL
tumor density
tumor maintenance
uterine sarcoma
xenograft
Xenopus laevis
XIAP antagonists
XIAP-BIR3 domain
yatein
α9-nAChR
β-glucans
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Altri titoli varianti Role of Natural Bioactive Compounds in the Rise and Fall of Cancers
Record Nr. UNINA-9910557476303321
Luparello Claudio  
Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2020
Materiale a stampa
Lo trovi qui: Univ. Federico II
Opac: Controlla la disponibilità qui
Synthesis, Study and Utilization of Natural Products
Synthesis, Study and Utilization of Natural Products
Autore Drasar Pavel B
Pubbl/distr/stampa MDPI - Multidisciplinary Digital Publishing Institute, 2020
Descrizione fisica 1 online resource (234 p.)
Soggetto topico Technology: general issues
Soggetto non controllato 4-epi-varioxiranol A
absolute structure
adhesive
anti-inflammation
anticancer drug
antioxidant
antioxidant activity
apo-CpcB
apoptosis
bardoxolone methyl
bioactivity
biosynthesis
bromelain
caffeoylquinic acids
cancer cells
cell opening
chlorogenic acid
cytotoxicity
derivatives
Emericella variecolor
fatty acid
flavonoids
flexible polyurethane foam
flow cytometry
gene expression
genetical transformation
ginkgolide
HepG2 cells
inhibitor
insect sex pheromone
isosorbide
lipid-lowering effects
live-cell fluorescence microscopy
melatonin
microbial biosynthesis
mitochondria
n/a
natural enantiomer
natural product
natural products
octadecanoid
oleic acid-elicited
PEGylated purpurin 18
pharmacokinetic features
pharmacological activities
phenolic acid
photodynamic therapy
photosensitizer
phototoxicity
phycocyanin
pinocembrin
Plantago depressa
platelet-activating factor receptor
polyphenol
polysaccharides
post-translationally modified peptides
radical scavenger
Ramulus mori
research progress
resource chemistry
reversible urethane linkages
rheumatoid arthritis
ribosomally synthesized
RiPP
salt stress
singlet oxygen
SlCOMT1
soy protein isolate
Spirulina
stilbene
synthesis of natural products
tea tussock moth
tomato
total synthesis
triglycidylamine
triterpenoids
varioxiranol A
viscosity
water resistance
ISBN 3-03928-153-4
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Record Nr. UNINA-9910372783503321
Drasar Pavel B  
MDPI - Multidisciplinary Digital Publishing Institute, 2020
Materiale a stampa
Lo trovi qui: Univ. Federico II
Opac: Controlla la disponibilità qui
Unconventional Anticancer Metallodrugs and Strategies to Improve their Pharmacological Profile / Maria Contel
Unconventional Anticancer Metallodrugs and Strategies to Improve their Pharmacological Profile / Maria Contel
Autore Contel Maria
Pubbl/distr/stampa MDPI - Multidisciplinary Digital Publishing Institute, 2019
Descrizione fisica 1 electronic resource (204 p.)
Soggetto topico Biology, life sciences
Soggetto non controllato ?-? stacking
encapsulation
oxindolimine-metal complexes
cyclodextrin
platinum iodido complexes
distribution coefficient
antiproliferative activity
anticancer agents
nanotubes
ruthenium
platinum
Log kw
nanoparticles
drug discovery
metal complex
metallodrugs
isatin-derived ligands
anticancer drug
upconverting nanoparticles
pyridine benzimidazole
dendrimers
liposomes
thiophene
angiogenesis
micelles
HSA oxidation
platinum(IV)
imaging
chromatographic lipophilicity parameter
amidophosphine
copper and iron chelators in cancer
Log P
biomacromolecules
bones
DNA cleavage
stopped-flow spectroscopy
silver
phosphonates
transmetalation
metallomics
MRI
fluorescence quenching
partition coefficient
gold fingers
anticancer
HSA binding
gold
?0
targeting
metastasis
DNA interaction
antimigration
cytotoxicity
HPLC
ruthenium complexes
zinc finger proteins
Gold(III) complexes
aquaporins
antiproliferative
protein-DNA recognition
photoactivation
lipophilicity
cancer
1-methylcytosine
PET
ISBN 9783039213160
3039213164
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Record Nr. UNINA-9910367755103321
Contel Maria  
MDPI - Multidisciplinary Digital Publishing Institute, 2019
Materiale a stampa
Lo trovi qui: Univ. Federico II
Opac: Controlla la disponibilità qui