Anticancer Agents : Design, Synthesis and Evaluation |
Autore | Chen Qiao-Hong |
Pubbl/distr/stampa | Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021 |
Descrizione fisica | 1 electronic resource (606 p.) |
Soggetto topico | Medicine |
Soggetto non controllato |
benzofurans
chemical synthesis cytotoxic properties HeLa MOLT-4 K562 anticancer anti-neuroinflammation coumarin dihydroartemisinin flavonoids allene E-stereoselective regioselective anti-cancer activity cyanopyridone substituted pyridine pyridotriazine pyrazolopyridine thioxotriazopyridine anticancer activity HepG2 antitumor activity computational docking MDM2-p53 interaction xanthones yeast-based assays estrone derivatives hydrazine N-substituted pyrazoline anti-ovarian cancer topoisomerase II inhibitor kinase inhibitor antiproliferative agent urea synthesis antiproliferative activity apoptosis indoleamine 2,3-dioxygenase inhibitor anti-tumor immune modulation tryptophan metabolism taxoids βIII-tubulin P-glycoprotein drug resistance thiopene thienopyrimidinone thiazolidinone breast cancer benzofuran–pyrazole nanoparticles cytotoxic activity PARP-1 inhibition 3,6-dibromocarbazole 5-bromoindole carbazole actin migration Thienopyrimidine Pyrazole PI3Kα inhibitor quinazolin-4(3H)-one quinazolin-4(3H)-thione Schiff base antioxidant activity DFT study ortho-quinones beta-lapachone tanshione IIA PI3Ks PI3Kδ inhibitors 2H-benzo[e][1,2,4]thiadiazine 1,1-dioxide anticancer agents protein–protein interactions virtual screening mimetics drug discovery bivalency polyvalency antitumor cell cycle ovarian cancer P-MAPA IL-12 TLR signaling inflammation chemoresistance 4-(pyridin-4-yloxy)benzamide 1,2,3-triazole c-Met natural product anticancer agent zampanolide Talazoparib PARP inhibitor prodrug o-nitro-benzyl photoactivatable protecting groups salinomycin overcoming drug resistance tumor specificity synergy 5-fluorouracil gemcitabine amides/esters colchicine analogs thiocolchicine colchiceine antimitotic agents hydrates dihydropyranoindole HDAC inhibitors neuroblastoma aromatase MCF-7 NIH3T3 benzimidazole triazolothiadiazine docking ADME organosilicon compounds SILA-409 (Alis-409) SILA-421 (Alis-421) multidrug resistance (MDR) reversal ABCB1 (P-glycoprotein) colon cancer colchicine amide colchicine sulfonamide tubulin inhibitors docking studies crystal structure PROTACs protein degradation IGF-1R Src protein kinase phenylpyrazolopyrimidine enzyme inhibition molecular simulation androgen receptor prostate cancer enzalutamide apalutamide darolutamide triple-negative breast cancer cytotoxicity chrysin analogues flavonoid anticancer compounds |
Formato | Materiale a stampa |
Livello bibliografico | Monografia |
Lingua di pubblicazione | eng |
Altri titoli varianti | Anticancer Agents |
Record Nr. | UNINA-9910557129103321 |
Chen Qiao-Hong | ||
Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021 | ||
Materiale a stampa | ||
Lo trovi qui: Univ. Federico II | ||
|
Bioactive Molecules from Extreme Environments |
Autore | Giordano Daniela (Researcher) |
Pubbl/distr/stampa | Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021 |
Descrizione fisica | 1 electronic resource (244 p.) |
Soggetto topico | Medicine |
Soggetto non controllato |
Latrunculia
Antarctica deep-sea sponge molecular networking molecular docking discorhabdin Arctic/Antarctic environment biocatalysis cold-adaptation marine biotechnology deep sea extremophilic microorganisms extremozyme thermophilic enzyme psychrophilic enzyme halophilic enzyme piezophilic enzyme chitinase cold-adapted optimization antifungal Pseudomonas Deinococcus deinoxanthin carotenoid deep-sea extreme ecosystem fungi bioactive compounds secondary metabolites halophilic bacteria archaea and fungi biomolecules biomedicine antimicrobial compounds anticancer compounds green synthesis biomaterials silver nitrate antibiotics nanotechnology marine prokaryotes microbial diversity polyextremophiles deep hypersaline anoxic basins blue biotechnologies extremozymes limits of life Antarctic krill (Euphausia superba) genome survey mitochondrial genome whiteleg shrimp (Penaeus vannamei) antimicrobial peptide (AMP) antihypertensive peptide (AHTP) cypermethrin biosurfactants biodegradation capacities marine sediments Arctic/Antarctic deep hypersaline anoxic basin cold-adapted bacteria halophilic microorganisms marine natural product enzyme silver nanoparticle marine bioprospecting |
Formato | Materiale a stampa |
Livello bibliografico | Monografia |
Lingua di pubblicazione | eng |
Record Nr. | UNINA-9910557147603321 |
Giordano Daniela (Researcher) | ||
Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021 | ||
Materiale a stampa | ||
Lo trovi qui: Univ. Federico II | ||
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Nanostructured Materials based on Noble Metals for Advanced Biological Applications |
Autore | Venditti Iole |
Pubbl/distr/stampa | Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2020 |
Descrizione fisica | 1 electronic resource (124 p.) |
Soggetto topico | Technology: general issues |
Soggetto non controllato |
gold
nanostructure EDTA tetrasodium salt photothermal therapy silver nanoparticles biomedical applications biological interactions biofunctional performances intrinsic anti-inflammatory activity antimicrobial efficiency localized surface plasmon resonance dip-coating capillary force exosome gold nanoparticles copper(I) complexes conjugates drug delivery anticancer compounds niosomes liposomes plasmonic materials nanocarriers Hg2+ sensors heavy metal sensing plasmonic sensors optical sensors ecosafety nanoparticles interactions protein corona nanomedicine biomolecules nanomaterials noble metal nanoparticles gold nanomaterials silver nanomaterials hybrid metal–polymer nanoparticles biotechnological applications nanomaterials for drug delivery nanomaterials for sensing |
Formato | Materiale a stampa |
Livello bibliografico | Monografia |
Lingua di pubblicazione | eng |
Record Nr. | UNINA-9910557641003321 |
Venditti Iole | ||
Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2020 | ||
Materiale a stampa | ||
Lo trovi qui: Univ. Federico II | ||
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