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Anticancer Agents : Design, Synthesis and Evaluation
Anticancer Agents : Design, Synthesis and Evaluation
Autore Chen Qiao-Hong
Pubbl/distr/stampa Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021
Descrizione fisica 1 electronic resource (606 p.)
Soggetto topico Medicine
Soggetto non controllato benzofurans
chemical synthesis
cytotoxic properties
HeLa
MOLT-4
K562
anticancer
anti-neuroinflammation
coumarin
dihydroartemisinin
flavonoids
allene
E-stereoselective
regioselective
anti-cancer activity
cyanopyridone
substituted pyridine
pyridotriazine
pyrazolopyridine
thioxotriazopyridine
anticancer activity
HepG2
antitumor activity
computational docking
MDM2-p53 interaction
xanthones
yeast-based assays
estrone derivatives
hydrazine
N-substituted pyrazoline
anti-ovarian cancer
topoisomerase II inhibitor
kinase inhibitor
antiproliferative agent
urea
synthesis
antiproliferative activity
apoptosis
indoleamine 2,3-dioxygenase
inhibitor
anti-tumor
immune modulation
tryptophan metabolism
taxoids
βIII-tubulin
P-glycoprotein
drug resistance
thiopene
thienopyrimidinone
thiazolidinone
breast cancer
benzofuran–pyrazole
nanoparticles
cytotoxic activity
PARP-1 inhibition
3,6-dibromocarbazole
5-bromoindole
carbazole
actin
migration
Thienopyrimidine
Pyrazole
PI3Kα inhibitor
quinazolin-4(3H)-one
quinazolin-4(3H)-thione
Schiff base
antioxidant activity
DFT study
ortho-quinones
beta-lapachone
tanshione IIA
PI3Ks
PI3Kδ inhibitors
2H-benzo[e][1,2,4]thiadiazine 1,1-dioxide
anticancer agents
protein–protein interactions
virtual screening
mimetics
drug discovery
bivalency
polyvalency
antitumor
cell cycle
ovarian cancer
P-MAPA
IL-12
TLR signaling
inflammation
chemoresistance
4-(pyridin-4-yloxy)benzamide
1,2,3-triazole
c-Met
natural product
anticancer agent
zampanolide
Talazoparib
PARP inhibitor
prodrug
o-nitro-benzyl
photoactivatable protecting groups
salinomycin
overcoming drug resistance
tumor specificity
synergy
5-fluorouracil
gemcitabine
amides/esters
colchicine analogs
thiocolchicine
colchiceine
antimitotic agents
hydrates
dihydropyranoindole
HDAC inhibitors
neuroblastoma
aromatase
MCF-7
NIH3T3
benzimidazole
triazolothiadiazine
docking
ADME
organosilicon compounds
SILA-409 (Alis-409)
SILA-421 (Alis-421)
multidrug resistance (MDR) reversal
ABCB1 (P-glycoprotein)
colon cancer
colchicine amide
colchicine sulfonamide
tubulin inhibitors
docking studies
crystal structure
PROTACs
protein degradation
IGF-1R
Src
protein kinase
phenylpyrazolopyrimidine
enzyme inhibition
molecular simulation
androgen receptor
prostate cancer
enzalutamide
apalutamide
darolutamide
triple-negative breast cancer
cytotoxicity
chrysin analogues
flavonoid
anticancer compounds
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Altri titoli varianti Anticancer Agents
Record Nr. UNINA-9910557129103321
Chen Qiao-Hong  
Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021
Materiale a stampa
Lo trovi qui: Univ. Federico II
Opac: Controlla la disponibilità qui
Electrophilic additions to unsaturated systems / P. B. D. de la Mare, R. Bolton
Electrophilic additions to unsaturated systems / P. B. D. de la Mare, R. Bolton
Autore DE LA MARE, P. D. B.
Pubbl/distr/stampa Amsterdam [etc.] : Elsevier, 1982
Descrizione fisica XIII, 377 p. ; 24 cm
Disciplina 547.413
Collana Studies in organic chemistry
Soggetto non controllato acetilene - composti
allene
cumuleni
sintesi organica
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Record Nr. UNISA-990003296980203316
DE LA MARE, P. D. B.  
Amsterdam [etc.] : Elsevier, 1982
Materiale a stampa
Lo trovi qui: Univ. di Salerno
Opac: Controlla la disponibilità qui
Synthesis of acetylenes, allenes and cumulenes : a laboratory manual / L. Brandsma and H.D. Verkruijsse
Synthesis of acetylenes, allenes and cumulenes : a laboratory manual / L. Brandsma and H.D. Verkruijsse
Autore Brandsma, L.
Pubbl/distr/stampa Amsterdam [etc.] : Elsevier, 1981
Descrizione fisica IX, 276 p. ; 24 cm
Disciplina 547413
Collana Studies in organic chemistry
Soggetto non controllato acetilene - composti
allene
cumuleni
sintesi organica
ISBN 0-444-42009-6
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Record Nr. UNISA-990000235980203316
Brandsma, L.  
Amsterdam [etc.] : Elsevier, 1981
Materiale a stampa
Lo trovi qui: Univ. di Salerno
Opac: Controlla la disponibilità qui
Synthesis of acetylenes, allenes and cumulenes : a laboratory manual / L. Brandsma and H.D. Verkruijsse
Synthesis of acetylenes, allenes and cumulenes : a laboratory manual / L. Brandsma and H.D. Verkruijsse
Autore Brandsma, L.
Pubbl/distr/stampa Amsterdam [etc.] : Elsevier, 1981
Descrizione fisica IX, 276 p. ; 24 cm
Disciplina 547413
Collana Studies in organic chemistry
Soggetto non controllato acetilene - composti
allene
cumuleni
sintesi organica
ISBN 0-444-42009-6
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Record Nr. UNISA-990000129320203316
Brandsma, L.  
Amsterdam [etc.] : Elsevier, 1981
Materiale a stampa
Lo trovi qui: Univ. di Salerno
Opac: Controlla la disponibilità qui