Anticancer Agents : Design, Synthesis and Evaluation
| Anticancer Agents : Design, Synthesis and Evaluation |
| Autore | Chen Qiao-Hong |
| Pubbl/distr/stampa | Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021 |
| Descrizione fisica | 1 online resource (606 p.) |
| Soggetto topico | Medicine and Nursing |
| Soggetto non controllato |
1,2,3-triazole
2H-benzo[e][1,2,4]thiadiazine 1,1-dioxide 3,6-dibromocarbazole 4-(pyridin-4-yloxy)benzamide 5-bromoindole 5-fluorouracil ABCB1 (P-glycoprotein) actin ADME allene amides/esters androgen receptor anti-cancer activity anti-neuroinflammation anti-ovarian cancer anti-tumor anticancer anticancer activity anticancer agent anticancer agents anticancer compounds antimitotic agents antioxidant activity antiproliferative activity antiproliferative agent antitumor antitumor activity apalutamide apoptosis aromatase benzimidazole benzofuran-pyrazole benzofurans beta-lapachone bivalency breast cancer c-Met carbazole cell cycle chemical synthesis chemoresistance chrysin analogues colchiceine colchicine amide colchicine analogs colchicine sulfonamide colon cancer computational docking coumarin crystal structure cyanopyridone cytotoxic activity cytotoxic properties cytotoxicity darolutamide DFT study dihydroartemisinin dihydropyranoindole docking docking studies drug discovery drug resistance E-stereoselective enzalutamide enzyme inhibition estrone derivatives flavonoid flavonoids gemcitabine HDAC inhibitors HeLa HepG2 hydrates hydrazine IGF-1R IL-12 immune modulation indoleamine 2,3-dioxygenase inflammation inhibitor K562 kinase inhibitor MCF-7 MDM2-p53 interaction migration mimetics molecular simulation MOLT-4 multidrug resistance (MDR) reversal N-substituted pyrazoline nanoparticles natural product neuroblastoma NIH3T3 o-nitro-benzyl organosilicon compounds ortho-quinones ovarian cancer overcoming drug resistance P-glycoprotein P-MAPA PARP inhibitor PARP-1 inhibition phenylpyrazolopyrimidine photoactivatable protecting groups PI3Ks PI3Kα inhibitor PI3Kδ inhibitors polyvalency prodrug prostate cancer PROTACs protein degradation protein kinase protein-protein interactions Pyrazole pyrazolopyridine pyridotriazine quinazolin-4(3H)-one quinazolin-4(3H)-thione regioselective salinomycin Schiff base SILA-409 (Alis-409) SILA-421 (Alis-421) Src substituted pyridine synergy synthesis Talazoparib tanshione IIA taxoids thiazolidinone Thienopyrimidine thienopyrimidinone thiocolchicine thiopene thioxotriazopyridine TLR signaling topoisomerase II inhibitor triazolothiadiazine triple-negative breast cancer tryptophan metabolism tubulin inhibitors tumor specificity urea virtual screening xanthones yeast-based assays zampanolide βIII-tubulin |
| Formato | Materiale a stampa |
| Livello bibliografico | Monografia |
| Lingua di pubblicazione | eng |
| Altri titoli varianti | Anticancer Agents |
| Record Nr. | UNINA-9910557129103321 |
Chen Qiao-Hong
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| Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021 | ||
| Lo trovi qui: Univ. Federico II | ||
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Biological and Pharmacological Activity of Plant Natural Compounds II
| Biological and Pharmacological Activity of Plant Natural Compounds II |
| Autore | Pezzani Raffaele |
| Pubbl/distr/stampa | Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022 |
| Descrizione fisica | 1 online resource (338 p.) |
| Soggetto topico |
Medicine and Nursing
Pharmacology |
| Soggetto non controllato |
70% partial hepatectomy
actin polymerization advanced glycation end product (AGE) AGE-inhibitor anti-cancer anti-diabetic drugs anti-inflammatory activity anti-urolithiatic activity antidiabetic antidiabetic activity antimicrobial and anticancer activities antioxidant antioxidant activity antioxidants apoptosis Aquilaria sinensis Astragali Radix astragaloside IV Astragalus membranaceus Bergenia species bergenin Biebersteinia heterostemon botanical description brain-derived neurotrophic factor breast cancer Caenorhabditis elegans Callicarpa longissima carnosol chlorogenic acid Clerodendrum infortunatum coffee Combretum indicum L. cyclooxygenase cytotoxicity DAF-16 detoxification ability diabetes mellitus diabetic nephropathy Diclofenac dorsal hippocampus formation epithelial to mesenchymal transition espresso ethylene glycol Flaxseed oil galegine Ginkgo biloba glioblastoma HeLA cells hepatoprotection HepG-2 cells histopathology histophatology HT-1080 huang qi hypotensive immunomodulatory effect instant coffee LC-ESI-MS/MS leaf extract linusorb B3 liver liver regeneration MCF-7 MDA memory methylcellulose MMP-2 MMP-9 monoterpenes nano-emulsion network pharmacology neuroprotection object recognition Ostrich oil oxidative stress Peganum harmala pharmacology phenylpropanoids pheophorbide A phytochemistry platelet aggregation polyphenols proliferation rat rheumatoid arthritis rosmanol Rubia tinctorum L. Saccharomyces cerevisiae Sage Salvia officinalis Src Struthio camelus swertiamarin synergistic effect TAOxC terpenoids TLR4/NF-κB/MAPK toxicity traditional medicine traditional uses UPLC-QTOF/ESI-MS urolithiasis β-glucan γ-lactone |
| Formato | Materiale a stampa |
| Livello bibliografico | Monografia |
| Lingua di pubblicazione | eng |
| Record Nr. | UNINA-9910566486603321 |
Pezzani Raffaele
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| Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022 | ||
| Lo trovi qui: Univ. Federico II | ||
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Theme Issue Honoring Prof. Dr. Ludger Wessjohann’s 60th Birthday: Natural Products in Modern Drug Discovery
| Theme Issue Honoring Prof. Dr. Ludger Wessjohann’s 60th Birthday: Natural Products in Modern Drug Discovery |
| Autore | Hussain Hidayat |
| Pubbl/distr/stampa | Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022 |
| Descrizione fisica | 1 online resource (360 p.) |
| Soggetto topico |
Chemistry
Organic chemistry Research and information: general |
| Soggetto non controllato |
ampullosporin
angiogenesis anti-tumor peptides antibody engineering anticancer anticancer activity antifungal antiproliferative apoptosis apoptosis resistance ATG 4B biorthogonal chemistry bispecific antibody botanical agents breast cancer butein cancer stem cells cancer treatment caspase-3 click chemistry co-culture coronavirus Cosmospora sp COX inhibitory cytotoxic cytotoxic activity DARTS Decachaeta incompta demissidine docking drug resistance ECD-TDDFT electron paramagnetic resonance (EPR) spectroscopy flavonoids frondoside-A fusidic acid glutamic acid methyl ester hepatocellular carcinoma in vitro model incomptine A invasion iTRAQ kaempferol lung cancer Magnaporthe oryzae marine fungi medicinal herbs melanoma MERS-CoV metabolomics metastasis molecular docking molecular networking multi-component reaction n/a natural products ophiobolin A PCD peptaibols phytochemicals phytopathogen polygodial pregnancy proliferation RCE-4 ROS production SARS-CoV SARS-CoV-2 Sepedonium ampullosporum sesquiterpene lactone solanidane alkaloids solanidine solid-phase peptide synthesis soudanone Sparticola junci Src STAT3 stemness steroidal alkaloids structure elucidation target identification TEMPO-conjugate the Bcl-2-Beclin 1 complex Trypsiligase tumor growth tumor heterogeneity tumor microenvironment (TME) viability violacein Wittig reaction |
| Formato | Materiale a stampa |
| Livello bibliografico | Monografia |
| Lingua di pubblicazione | eng |
| Altri titoli varianti | Theme Issue Honoring Prof. Dr. Ludger Wessjohann’s 60th Birthday |
| Record Nr. | UNINA-9910585945403321 |
Hussain Hidayat
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| Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022 | ||
| Lo trovi qui: Univ. Federico II | ||
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