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Anticancer Agents : Design, Synthesis and Evaluation
Anticancer Agents : Design, Synthesis and Evaluation
Autore Chen Qiao-Hong
Pubbl/distr/stampa Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021
Descrizione fisica 1 online resource (606 p.)
Soggetto topico Medicine and Nursing
Soggetto non controllato 1,2,3-triazole
2H-benzo[e][1,2,4]thiadiazine 1,1-dioxide
3,6-dibromocarbazole
4-(pyridin-4-yloxy)benzamide
5-bromoindole
5-fluorouracil
ABCB1 (P-glycoprotein)
actin
ADME
allene
amides/esters
androgen receptor
anti-cancer activity
anti-neuroinflammation
anti-ovarian cancer
anti-tumor
anticancer
anticancer activity
anticancer agent
anticancer agents
anticancer compounds
antimitotic agents
antioxidant activity
antiproliferative activity
antiproliferative agent
antitumor
antitumor activity
apalutamide
apoptosis
aromatase
benzimidazole
benzofuran-pyrazole
benzofurans
beta-lapachone
bivalency
breast cancer
c-Met
carbazole
cell cycle
chemical synthesis
chemoresistance
chrysin analogues
colchiceine
colchicine amide
colchicine analogs
colchicine sulfonamide
colon cancer
computational docking
coumarin
crystal structure
cyanopyridone
cytotoxic activity
cytotoxic properties
cytotoxicity
darolutamide
DFT study
dihydroartemisinin
dihydropyranoindole
docking
docking studies
drug discovery
drug resistance
E-stereoselective
enzalutamide
enzyme inhibition
estrone derivatives
flavonoid
flavonoids
gemcitabine
HDAC inhibitors
HeLa
HepG2
hydrates
hydrazine
IGF-1R
IL-12
immune modulation
indoleamine 2,3-dioxygenase
inflammation
inhibitor
K562
kinase inhibitor
MCF-7
MDM2-p53 interaction
migration
mimetics
molecular simulation
MOLT-4
multidrug resistance (MDR) reversal
N-substituted pyrazoline
nanoparticles
natural product
neuroblastoma
NIH3T3
o-nitro-benzyl
organosilicon compounds
ortho-quinones
ovarian cancer
overcoming drug resistance
P-glycoprotein
P-MAPA
PARP inhibitor
PARP-1 inhibition
phenylpyrazolopyrimidine
photoactivatable protecting groups
PI3Ks
PI3Kα inhibitor
PI3Kδ inhibitors
polyvalency
prodrug
prostate cancer
PROTACs
protein degradation
protein kinase
protein-protein interactions
Pyrazole
pyrazolopyridine
pyridotriazine
quinazolin-4(3H)-one
quinazolin-4(3H)-thione
regioselective
salinomycin
Schiff base
SILA-409 (Alis-409)
SILA-421 (Alis-421)
Src
substituted pyridine
synergy
synthesis
Talazoparib
tanshione IIA
taxoids
thiazolidinone
Thienopyrimidine
thienopyrimidinone
thiocolchicine
thiopene
thioxotriazopyridine
TLR signaling
topoisomerase II inhibitor
triazolothiadiazine
triple-negative breast cancer
tryptophan metabolism
tubulin inhibitors
tumor specificity
urea
virtual screening
xanthones
yeast-based assays
zampanolide
βIII-tubulin
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Altri titoli varianti Anticancer Agents
Record Nr. UNINA-9910557129103321
Chen Qiao-Hong  
Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021
Materiale a stampa
Lo trovi qui: Univ. Federico II
Opac: Controlla la disponibilità qui
Biological and Pharmacological Activity of Plant Natural Compounds II
Biological and Pharmacological Activity of Plant Natural Compounds II
Autore Pezzani Raffaele
Pubbl/distr/stampa Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022
Descrizione fisica 1 online resource (338 p.)
Soggetto topico Medicine and Nursing
Pharmacology
Soggetto non controllato 70% partial hepatectomy
actin polymerization
advanced glycation end product (AGE)
AGE-inhibitor
anti-cancer
anti-diabetic drugs
anti-inflammatory activity
anti-urolithiatic activity
antidiabetic
antidiabetic activity
antimicrobial and anticancer activities
antioxidant
antioxidant activity
antioxidants
apoptosis
Aquilaria sinensis
Astragali Radix
astragaloside IV
Astragalus membranaceus
Bergenia species
bergenin
Biebersteinia heterostemon
botanical description
brain-derived neurotrophic factor
breast cancer
Caenorhabditis elegans
Callicarpa longissima
carnosol
chlorogenic acid
Clerodendrum infortunatum
coffee
Combretum indicum L.
cyclooxygenase
cytotoxicity
DAF-16
detoxification ability
diabetes mellitus
diabetic nephropathy
Diclofenac
dorsal hippocampus formation
epithelial to mesenchymal transition
espresso
ethylene glycol
Flaxseed oil
galegine
Ginkgo biloba
glioblastoma
HeLA cells
hepatoprotection
HepG-2 cells
histopathology
histophatology
HT-1080
huang qi
hypotensive
immunomodulatory effect
instant coffee
LC-ESI-MS/MS
leaf extract
linusorb B3
liver
liver regeneration
MCF-7
MDA
memory
methylcellulose
MMP-2
MMP-9
monoterpenes
nano-emulsion
network pharmacology
neuroprotection
object recognition
Ostrich oil
oxidative stress
Peganum harmala
pharmacology
phenylpropanoids
pheophorbide A
phytochemistry
platelet aggregation
polyphenols
proliferation
rat
rheumatoid arthritis
rosmanol
Rubia tinctorum L.
Saccharomyces cerevisiae
Sage
Salvia officinalis
Src
Struthio camelus
swertiamarin
synergistic effect
TAOxC
terpenoids
TLR4/NF-κB/MAPK
toxicity
traditional medicine
traditional uses
UPLC-QTOF/ESI-MS
urolithiasis
β-glucan
γ-lactone
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Record Nr. UNINA-9910566486603321
Pezzani Raffaele  
Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022
Materiale a stampa
Lo trovi qui: Univ. Federico II
Opac: Controlla la disponibilità qui
Theme Issue Honoring Prof. Dr. Ludger Wessjohann’s 60th Birthday: Natural Products in Modern Drug Discovery
Theme Issue Honoring Prof. Dr. Ludger Wessjohann’s 60th Birthday: Natural Products in Modern Drug Discovery
Autore Hussain Hidayat
Pubbl/distr/stampa Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022
Descrizione fisica 1 online resource (360 p.)
Soggetto topico Chemistry
Organic chemistry
Research and information: general
Soggetto non controllato ampullosporin
angiogenesis
anti-tumor peptides
antibody engineering
anticancer
anticancer activity
antifungal
antiproliferative
apoptosis
apoptosis resistance
ATG 4B
biorthogonal chemistry
bispecific antibody
botanical agents
breast cancer
butein
cancer stem cells
cancer treatment
caspase-3
click chemistry
co-culture
coronavirus
Cosmospora sp
COX inhibitory
cytotoxic
cytotoxic activity
DARTS
Decachaeta incompta
demissidine
docking
drug resistance
ECD-TDDFT
electron paramagnetic resonance (EPR) spectroscopy
flavonoids
frondoside-A
fusidic acid
glutamic acid methyl ester
hepatocellular carcinoma
in vitro model
incomptine A
invasion
iTRAQ
kaempferol
lung cancer
Magnaporthe oryzae
marine fungi
medicinal herbs
melanoma
MERS-CoV
metabolomics
metastasis
molecular docking
molecular networking
multi-component reaction
n/a
natural products
ophiobolin A
PCD
peptaibols
phytochemicals
phytopathogen
polygodial
pregnancy
proliferation
RCE-4
ROS production
SARS-CoV
SARS-CoV-2
Sepedonium ampullosporum
sesquiterpene lactone
solanidane alkaloids
solanidine
solid-phase peptide synthesis
soudanone
Sparticola junci
Src
STAT3
stemness
steroidal alkaloids
structure elucidation
target identification
TEMPO-conjugate
the Bcl-2-Beclin 1 complex
Trypsiligase
tumor growth
tumor heterogeneity
tumor microenvironment (TME)
viability
violacein
Wittig reaction
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Altri titoli varianti Theme Issue Honoring Prof. Dr. Ludger Wessjohann’s 60th Birthday
Record Nr. UNINA-9910585945403321
Hussain Hidayat  
Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022
Materiale a stampa
Lo trovi qui: Univ. Federico II
Opac: Controlla la disponibilità qui