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Anticancer Agents : Design, Synthesis and Evaluation
Anticancer Agents : Design, Synthesis and Evaluation
Autore Chen Qiao-Hong
Pubbl/distr/stampa Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021
Descrizione fisica 1 online resource (606 p.)
Soggetto topico Medicine and Nursing
Soggetto non controllato 1,2,3-triazole
2H-benzo[e][1,2,4]thiadiazine 1,1-dioxide
3,6-dibromocarbazole
4-(pyridin-4-yloxy)benzamide
5-bromoindole
5-fluorouracil
ABCB1 (P-glycoprotein)
actin
ADME
allene
amides/esters
androgen receptor
anti-cancer activity
anti-neuroinflammation
anti-ovarian cancer
anti-tumor
anticancer
anticancer activity
anticancer agent
anticancer agents
anticancer compounds
antimitotic agents
antioxidant activity
antiproliferative activity
antiproliferative agent
antitumor
antitumor activity
apalutamide
apoptosis
aromatase
benzimidazole
benzofuran-pyrazole
benzofurans
beta-lapachone
bivalency
breast cancer
c-Met
carbazole
cell cycle
chemical synthesis
chemoresistance
chrysin analogues
colchiceine
colchicine amide
colchicine analogs
colchicine sulfonamide
colon cancer
computational docking
coumarin
crystal structure
cyanopyridone
cytotoxic activity
cytotoxic properties
cytotoxicity
darolutamide
DFT study
dihydroartemisinin
dihydropyranoindole
docking
docking studies
drug discovery
drug resistance
E-stereoselective
enzalutamide
enzyme inhibition
estrone derivatives
flavonoid
flavonoids
gemcitabine
HDAC inhibitors
HeLa
HepG2
hydrates
hydrazine
IGF-1R
IL-12
immune modulation
indoleamine 2,3-dioxygenase
inflammation
inhibitor
K562
kinase inhibitor
MCF-7
MDM2-p53 interaction
migration
mimetics
molecular simulation
MOLT-4
multidrug resistance (MDR) reversal
N-substituted pyrazoline
nanoparticles
natural product
neuroblastoma
NIH3T3
o-nitro-benzyl
organosilicon compounds
ortho-quinones
ovarian cancer
overcoming drug resistance
P-glycoprotein
P-MAPA
PARP inhibitor
PARP-1 inhibition
phenylpyrazolopyrimidine
photoactivatable protecting groups
PI3Ks
PI3Kα inhibitor
PI3Kδ inhibitors
polyvalency
prodrug
prostate cancer
PROTACs
protein degradation
protein kinase
protein-protein interactions
Pyrazole
pyrazolopyridine
pyridotriazine
quinazolin-4(3H)-one
quinazolin-4(3H)-thione
regioselective
salinomycin
Schiff base
SILA-409 (Alis-409)
SILA-421 (Alis-421)
Src
substituted pyridine
synergy
synthesis
Talazoparib
tanshione IIA
taxoids
thiazolidinone
Thienopyrimidine
thienopyrimidinone
thiocolchicine
thiopene
thioxotriazopyridine
TLR signaling
topoisomerase II inhibitor
triazolothiadiazine
triple-negative breast cancer
tryptophan metabolism
tubulin inhibitors
tumor specificity
urea
virtual screening
xanthones
yeast-based assays
zampanolide
βIII-tubulin
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Altri titoli varianti Anticancer Agents
Record Nr. UNINA-9910557129103321
Chen Qiao-Hong  
Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021
Materiale a stampa
Lo trovi qui: Univ. Federico II
Opac: Controlla la disponibilità qui
Novel Anti-cancer Agents and Cellular Targets and Their Mechanism(s) of Action
Novel Anti-cancer Agents and Cellular Targets and Their Mechanism(s) of Action
Autore Allison Simon J
Pubbl/distr/stampa MDPI - Multidisciplinary Digital Publishing Institute, 2022
Descrizione fisica 1 online resource (206 p.)
Soggetto topico History of engineering & technology
Technology: general issues
Soggetto non controllato 5-FU resistance
8-hydroxydaidzein
affibody drug conjugate (AffiDC)
affibody molecule
albumin binding domain
angiogenesis
anti-cancer agent
anticancer drug
apoptosis
AQ4N
autophagy
B-lactam steroid alkylators
BCR-ABL
biomarker
bioprecursor
breast cancer
BxPC-3
c-myc
cancer hallmarks
CCN1
colorectal cancer
Connectivity Map
CYP1A1
CYP1B1
CYP2W1
Cytochrome P450
DM1
drug repurposing
duocarmycin
EGFR tyrosine kinase inhibitor
emtansine
expression
gene silencing
Genomics of Drug Sensitivity in Cancer
glioblastoma
HepG2
Huh7
human epidermal growth factor receptor 3 (HER3)
hybrid steroidal alkylating agents
in vivo imaging
invasion
isatin sulfonamides
K562
MAPK
mesenchymal-amoeboid transition
microtubule acetylation
migration
molecular docking
n/a
nanoparticles
nanosystems
NF-κB
oncogene
ovarian cancer
phortress
photon upconversion
PLGA
poly (ADP-ribose) polymerase inhibitors
prodrug
RNA interference
siRNA
synthetic lethality
triple-negative breast cancer
triplet-triplet annihilation
ISBN 3-0365-5222-7
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Altri titoli varianti Novel Anti-cancer Agents and Cellular Targets and Their Mechanism
Record Nr. UNINA-9910619465503321
Allison Simon J  
MDPI - Multidisciplinary Digital Publishing Institute, 2022
Materiale a stampa
Lo trovi qui: Univ. Federico II
Opac: Controlla la disponibilità qui