Anticancer Agents : Design, Synthesis and Evaluation
| Anticancer Agents : Design, Synthesis and Evaluation |
| Autore | Chen Qiao-Hong |
| Pubbl/distr/stampa | Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021 |
| Descrizione fisica | 1 online resource (606 p.) |
| Soggetto topico | Medicine and Nursing |
| Soggetto non controllato |
1,2,3-triazole
2H-benzo[e][1,2,4]thiadiazine 1,1-dioxide 3,6-dibromocarbazole 4-(pyridin-4-yloxy)benzamide 5-bromoindole 5-fluorouracil ABCB1 (P-glycoprotein) actin ADME allene amides/esters androgen receptor anti-cancer activity anti-neuroinflammation anti-ovarian cancer anti-tumor anticancer anticancer activity anticancer agent anticancer agents anticancer compounds antimitotic agents antioxidant activity antiproliferative activity antiproliferative agent antitumor antitumor activity apalutamide apoptosis aromatase benzimidazole benzofuran-pyrazole benzofurans beta-lapachone bivalency breast cancer c-Met carbazole cell cycle chemical synthesis chemoresistance chrysin analogues colchiceine colchicine amide colchicine analogs colchicine sulfonamide colon cancer computational docking coumarin crystal structure cyanopyridone cytotoxic activity cytotoxic properties cytotoxicity darolutamide DFT study dihydroartemisinin dihydropyranoindole docking docking studies drug discovery drug resistance E-stereoselective enzalutamide enzyme inhibition estrone derivatives flavonoid flavonoids gemcitabine HDAC inhibitors HeLa HepG2 hydrates hydrazine IGF-1R IL-12 immune modulation indoleamine 2,3-dioxygenase inflammation inhibitor K562 kinase inhibitor MCF-7 MDM2-p53 interaction migration mimetics molecular simulation MOLT-4 multidrug resistance (MDR) reversal N-substituted pyrazoline nanoparticles natural product neuroblastoma NIH3T3 o-nitro-benzyl organosilicon compounds ortho-quinones ovarian cancer overcoming drug resistance P-glycoprotein P-MAPA PARP inhibitor PARP-1 inhibition phenylpyrazolopyrimidine photoactivatable protecting groups PI3Ks PI3Kα inhibitor PI3Kδ inhibitors polyvalency prodrug prostate cancer PROTACs protein degradation protein kinase protein-protein interactions Pyrazole pyrazolopyridine pyridotriazine quinazolin-4(3H)-one quinazolin-4(3H)-thione regioselective salinomycin Schiff base SILA-409 (Alis-409) SILA-421 (Alis-421) Src substituted pyridine synergy synthesis Talazoparib tanshione IIA taxoids thiazolidinone Thienopyrimidine thienopyrimidinone thiocolchicine thiopene thioxotriazopyridine TLR signaling topoisomerase II inhibitor triazolothiadiazine triple-negative breast cancer tryptophan metabolism tubulin inhibitors tumor specificity urea virtual screening xanthones yeast-based assays zampanolide βIII-tubulin |
| Formato | Materiale a stampa |
| Livello bibliografico | Monografia |
| Lingua di pubblicazione | eng |
| Altri titoli varianti | Anticancer Agents |
| Record Nr. | UNINA-9910557129103321 |
Chen Qiao-Hong
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| Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021 | ||
| Lo trovi qui: Univ. Federico II | ||
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From Basic Research to New Tools and Challenges for the Genotoxicity Testing of Nanomaterials
| From Basic Research to New Tools and Challenges for the Genotoxicity Testing of Nanomaterials |
| Autore | FESSARD Valérie |
| Pubbl/distr/stampa | Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021 |
| Descrizione fisica | 1 online resource (188 p.) |
| Soggetto topico |
Humanities
Social interaction |
| Soggetto non controllato |
3D culture
advanced in vitro model AgNP Allium cepa aluminum antioxidant activity apoptosis BEAS-2B cells CeO2NP comet assay cytotoxic cytotoxicity DNA damage DNA methylation epigenetics FPG enzyme genotoxic genotoxicity graphene oxide gut hepatotoxicity HepG2 high throughput screening Hprt Hs27 human fibroblasts human amniotic cells in vitro genotoxicity in vitro testing lincomycin liver liver spheroids metal oxides metal/coating agent ratio micronuclei formation micronucleus micronucleus assay multi-walled carbon nanotubes (MWCNT) n/a nanomaterial nanoparticles nanoplastics nanotoxicology nongenotoxic silver nanoparticles oral route oxidative stress polystyrene nanoparticles reduced graphene oxide safer-by-design silver ions SiO2NP TiO2NP titanium dioxide nanoparticles tritiated particles tungsten V79 cells ZnONP |
| Formato | Materiale a stampa |
| Livello bibliografico | Monografia |
| Lingua di pubblicazione | eng |
| Record Nr. | UNINA-9910557414003321 |
FESSARD Valérie
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| Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021 | ||
| Lo trovi qui: Univ. Federico II | ||
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Functional Cereal Foods for Health Benefits: Genetic and/or Processing Strategies to Enhance the Quali-Quantitative Composition of Bioactive Components
| Functional Cereal Foods for Health Benefits: Genetic and/or Processing Strategies to Enhance the Quali-Quantitative Composition of Bioactive Components |
| Autore | Laddomada Barbara |
| Pubbl/distr/stampa | Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022 |
| Descrizione fisica | 1 online resource (228 p.) |
| Soggetto topico |
Biology, life sciences
Research and information: general |
| Soggetto non controllato |
air classification
air-classification plant air-classified fractions alveographic properties anti-atherogenic anti-diabetic anti-inflammatory anti-proliferative antioxidant antioxidant activity antioxidants apoptosis arsenic artificial neural network (ANN) ATI bound phenolic breadmaking buckwheat Caco-2 celiac disease cell cycle analysis cell growth inhibition climate constraints coix seed dehulling dietary fiber durum grains durum wheat enzymes fermentation free phenolic genetic variability germination gluten gluten strength glutenins grain protein content haplotypes HEp2 HepG2 heritability inorganic contaminants LC-MS leavened pancake maize inbred lines micronization plant milled rice milling fractions milling methods Monascus purpureus multiple linear regression (MLR) mycotoxins n/a non-celiac wheat/gluten sensitivity nutrients nutritional value organic contaminants phenolic acid phenolic compounds protein quality SNPs sorghum sorghum phenolics starch steamed bread Triticum aestivum L. Triticum durum Desf wheat wheat allergy yield performance |
| Formato | Materiale a stampa |
| Livello bibliografico | Monografia |
| Lingua di pubblicazione | eng |
| Altri titoli varianti | Functional Cereal Foods for Health Benefits |
| Record Nr. | UNINA-9910585944403321 |
Laddomada Barbara
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| Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022 | ||
| Lo trovi qui: Univ. Federico II | ||
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New Advances in the Research of Antioxidant Food Peptides
| New Advances in the Research of Antioxidant Food Peptides |
| Autore | Amigo Lourdes |
| Pubbl/distr/stampa | Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021 |
| Descrizione fisica | 1 online resource (154 p.) |
| Soggetto topico | Research and information: general |
| Soggetto non controllato |
aged animals
albumin albumin peptide animal protein antioxidant antioxidant activity antioxidant enzymes antioxidant peptide antioxidant peptides bioactive peptide bioactive peptides C2C12 cell models cellular ROS egg white egg yolk exercise extraction food antioxidant food peptides fruit residues HepG2 hydrolysis condition in silico multifunctionality mung bean mung bean albumin muscle n/a older adult ORAC peptide sequencing peptides reactive oxygen species sarcopenia Vigna radiata whey protein whey protein hydrolysate |
| Formato | Materiale a stampa |
| Livello bibliografico | Monografia |
| Lingua di pubblicazione | eng |
| Record Nr. | UNINA-9910557793003321 |
Amigo Lourdes
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| Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021 | ||
| Lo trovi qui: Univ. Federico II | ||
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Novel Anti-cancer Agents and Cellular Targets and Their Mechanism(s) of Action
| Novel Anti-cancer Agents and Cellular Targets and Their Mechanism(s) of Action |
| Autore | Allison Simon J |
| Pubbl/distr/stampa | MDPI - Multidisciplinary Digital Publishing Institute, 2022 |
| Descrizione fisica | 1 online resource (206 p.) |
| Soggetto topico |
History of engineering & technology
Technology: general issues |
| Soggetto non controllato |
5-FU resistance
8-hydroxydaidzein affibody drug conjugate (AffiDC) affibody molecule albumin binding domain angiogenesis anti-cancer agent anticancer drug apoptosis AQ4N autophagy B-lactam steroid alkylators BCR-ABL biomarker bioprecursor breast cancer BxPC-3 c-myc cancer hallmarks CCN1 colorectal cancer Connectivity Map CYP1A1 CYP1B1 CYP2W1 Cytochrome P450 DM1 drug repurposing duocarmycin EGFR tyrosine kinase inhibitor emtansine expression gene silencing Genomics of Drug Sensitivity in Cancer glioblastoma HepG2 Huh7 human epidermal growth factor receptor 3 (HER3) hybrid steroidal alkylating agents in vivo imaging invasion isatin sulfonamides K562 MAPK mesenchymal-amoeboid transition microtubule acetylation migration molecular docking n/a nanoparticles nanosystems NF-κB oncogene ovarian cancer phortress photon upconversion PLGA poly (ADP-ribose) polymerase inhibitors prodrug RNA interference siRNA synthetic lethality triple-negative breast cancer triplet-triplet annihilation |
| ISBN | 3-0365-5222-7 |
| Formato | Materiale a stampa |
| Livello bibliografico | Monografia |
| Lingua di pubblicazione | eng |
| Altri titoli varianti | Novel Anti-cancer Agents and Cellular Targets and Their Mechanism |
| Record Nr. | UNINA-9910619465503321 |
Allison Simon J
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| MDPI - Multidisciplinary Digital Publishing Institute, 2022 | ||
| Lo trovi qui: Univ. Federico II | ||
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Plant Essential Oil with Biological Activity
| Plant Essential Oil with Biological Activity |
| Autore | Elshafie Hazem Salaheldin |
| Pubbl/distr/stampa | Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022 |
| Descrizione fisica | 1 online resource (264 p.) |
| Soggetto topico |
Medicine and Nursing
Pharmacology |
| Soggetto non controllato |
Aerva javanica
agri-food industry allelopathy angustione Anisosciadium lanatum Annona cherimola anti-inflammation anti-senility antibacterial antibacterial activity anticholinesterase activity antifungal activity antimicrobial antimicrobial activity antioxidant antioxidant activity antioxidant enzymes antioxidants apoptotic markers aromatic plants Asteraceae BCL-2 bioherbicides biological control Campylobacter jejuni CASPASE-3 cell membrane permeability chemical composition chemometric analysis chemotype Cleome genus Curcuma longa cytotoxicity damage index eco-friendly product Ecuador enantiomers enantioselective analysis environmental factors essential oil essential oils extraction methods food preservatives fruit storage Fusarium root rot GC-MS germacrene D green chemistry HepG2 herbicidal herbicides horseweed hydrodistillation Jungia bullata Jungia jelskii Jungia malvifolia Jungia rugosa medicinal plants Mentha longifolia GC-MS Mentha spicata natural products Oncosiphon suffruticosum pale smartweed phytopathogens phytotoxicity postharvest diseases Pulicaria crispa quality preservation quality-related attributes sandy soil seasonal variation sesquiterpenes sun protection factor terpenes tomato trichomes tyrosinase inhibition volatile oils volatiles wavy-leaf fleabane WRKY transcription factor |
| Formato | Materiale a stampa |
| Livello bibliografico | Monografia |
| Lingua di pubblicazione | eng |
| Record Nr. | UNINA-9910566457203321 |
Elshafie Hazem Salaheldin
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| Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022 | ||
| Lo trovi qui: Univ. Federico II | ||
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