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From a Molecule to a Drug: Chemical Features Enhancing Pharmacological Potential
From a Molecule to a Drug: Chemical Features Enhancing Pharmacological Potential
Autore Ribaudo Giovanni
Pubbl/distr/stampa Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022
Descrizione fisica 1 electronic resource (234 p.)
Soggetto topico Medicine
Pharmacology
Soggetto non controllato SARS-CoV-2
benzoic acid derivatives
gallic acid
molecular docking
reactivity parameters
selenoxide elimination
one-pot
imine-enamine
reaction mechanism
DFT calculations
selenium
anti-inflammatory drugs
QSAR
pain management
cyclooxygenase
multitarget drug
cannabinoid
neuropathic pain
clopidogrel
NMR study
oxone
peroxymonosulfate
sodium halide
thienopyridine
drug discovery
precision medicine
pharmacodynamics
pharmacokinetics
coronavirus SARS-CoV-2
COVID-19
3-chymotrypsin-like protease
pyrimidonic pharmaceuticals
molecular dynamics simulations
binding free energy
β-carrageenan
antioxidant activity
Box-Behken
extraction
Eucheuma gelatinae
physic-chemistry
rheology
quercetin
quercetin 3-O-glucuronide
cisplatin
nephrotoxicity
cytoprotection
lithium therapy
neurocytology
toxicology
neuroprotection
chemoinformatics
big data
methadone hydrochloride
pharmaceutical solutions
drug compounding
high performance liquid chromatography
stability study
microbiology
fucoidan
alginate
L-selectin
E-selectin
MCP-1
ICAM-1
THP-1 macrophage
monocyte migration
protein binding
breast milk
M/P ratio
statistical modeling
molecular descriptors
chromatographic descriptors
affinity chromatography
anti-ACE
anti-DPP-IV
gastrointestinal digestion
in silico
molecular dynamics
paramyosin
seafood
target fishing
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Altri titoli varianti From a Molecule to a Drug
Record Nr. UNINA-9910585940503321
Ribaudo Giovanni  
Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022
Materiale a stampa
Lo trovi qui: Univ. Federico II
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Marine Drug Research in China: Selected Papers from the 15-NASMD Conference
Marine Drug Research in China: Selected Papers from the 15-NASMD Conference
Autore Zhou Xuefeng
Pubbl/distr/stampa Basel, : MDPI Books, 2022
Descrizione fisica 1 electronic resource (512 p.)
Soggetto topico Medicine
Soggetto non controllato Antarctic krill (Euphausia superba)
peptide
antioxidant activity
stability
oyster
plasma
peptidome
antimicrobial peptides
cytotoxicity
actinomycete
piericidins
absolute configuration
Pestalotiopsis heterocornis
heterocornols
anti-inflammatory activity
sponge-derived fungus
sclerotides
lipodepsipeptide
Aspergillus sclerotiorum
nasopharyngeal carcinoma
AChE inhibitory
vascular endothelial cell
flavonoid
oxidized low-density lipoprotein
Nrf2
apoptosis
butyrolactone I
food allergy
metabolism
pharmacokinetics
actinomycin X2
microbial pigments
dyeing
silk
antibacterial properties
PD-L1
virtual screening
pharmacophore modeling
ADME
molecular dynamics
xanthones
ascidian-derived fungus
Diaporthe sp
anti-glioma activity
antiaging
Sonneratia apetala
signaling pathway
Caenorhabditis elegans
mutants
coral-derived fungi
Aspergillus hiratsukae
meroterpenoids
antibacterial activity
cytotoxic activity
deep-sea-derived fungus
Aspergillus puniceus
isoquinoline alkaloid
protein tyrosine phosphatase inhibitor
antibacterial
Aspergillus sp
geodin
semisynthesize
insecticidal activity
Arca inflata
antitumor peptide
MAPK signaling
calmodulin
colorectal cancer
methicillin-resistant Staphylococcus aureus
actinomycin D
Streptomyces parvulus
mechanism
mangrove endophytic Pestalotiopsis
Sdy-1
antitumor activity
Wnt signaling
β-catenin
eremophilane sesquiterpenoids
mangrove-derived fungus
Penicillium sp
Oceanapia
sponge
secondary metabolites
biological activities
drug design
anticancer
cyclic pentapeptide
galaxamide analogues
skipjack tuna (Katsuwonus pelamis) muscle
angiotensin-I-converting enzyme (ACE) peptide
molecular docking
nitric oxide (NO)
endothelin-1 (ET-1)
Trichoderma longibrachiatum
sesquiterpene glycoside
antimicrobial activity
marine fungi
Aspergillus unguis
depsides
depsidones
osteoclast differentiation
soft-coral-derived fungus
pyranodipyran derivatives
tyrosyl DNA phosphodiesterase 1 inhibitory activities
fluorescent properties
butenolides
enantiomers
Aspergillus terreus
pancreatic lipase
NAFLD
fucoxanthin
adenosine monophosphate-activated protein kinase (AMPK)
nuclear factor erythroid-2-related factor 2-mediated (Nrf2)
Toll-like receptor 4-mediated (TLR4)
Aspergillus flavipes HN4-13
emodin
macroporous resin XAD-16
adsorption kinetics and isotherms
enrichment
tetramic acid derivatives
deep-sea fungus
clavipitacae
Lecanicillium fusisporum
chronic kidney disease
fucoidan
cognitive dysfunction
neuroinflammation
oxidative stress
GSK3β-Nrf2-HO-1 signaling
microglial polarization
deep-sea actinomycetes
aromatic acids
oximes
antihyperlipidemic
phycocyanin
microbiota
transcriptome
IL-17 pathway
Hahella
prodiginine
chejuenlide
genome mining
LC-MS/MS
CDK4/6
marine compounds
pharmacophore construction
ADMET
mm-pbsa
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Altri titoli varianti Marine Drug Research in China
Record Nr. UNINA-9910595071903321
Zhou Xuefeng  
Basel, : MDPI Books, 2022
Materiale a stampa
Lo trovi qui: Univ. Federico II
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Micro/Nanofluidic and Lab-on-a-Chip Devices for Biomedical Applications
Micro/Nanofluidic and Lab-on-a-Chip Devices for Biomedical Applications
Autore Carvalho Violeta
Pubbl/distr/stampa Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022
Descrizione fisica 1 electronic resource (232 p.)
Soggetto topico Medicine
Soggetto non controllato protein biomarker
microarray
microfluidic cassette
multiplex measurement
immunoassay
point-of-care testing
microfluidic device
small intestine
ex vivo
histology
embedded resin
sectioning
peptide biosensor
lab-on-a-chip
label-free detection
peptide aptamers
protein biomarkers
microfluidic biochip
troponin T
computational simulations
drug discovery
organ-on-a-chip
microfluidic devices
preclinical models
numerical simulations
automation
non-enzymatic
DNA amplification
L-DNA
microfluidic
fluorescence
paper microfluidics
sweat
sensing
hydrogels
lactate
osmotic pumping
evaporation
capillary
wicking
biochemical assay
microfluidics
cell trap
RBC
evolutionary algorithm
generative design
artificial intelligence
organ-on-chip
liver-on-chip
liver disease
multi-level microfluidic device
live cell imaging
long-term microscopy imaging
focus drifting
immersion oil viscosity
bacterial population dynamics
single-cell studies
E. coli
mother machine
computational fluid dynamics
cancer-on-chip
xenograft
colorectal cancer
pharmacodynamics
pharmacokinetics
drug efficacy
oxaliplatin
microfabrication
microphysiological system
biophysical stimuli
biochemical stimuli
in vitro cell culture
cortical neurons
hippocampal neurons
electrical stimulation
Micro-Electrode Arrays
engineered neuronal networks
polydimethylsiloxane
microchannels
in vivo micro bioreactor
additive manufacturing
poly-(ethylene glycol)-diacrylate
biocompatibility
COVID-19
diagnosis
image analysis
PCR
SARS-CoV-2
ISBN 3-0365-6099-8
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Record Nr. UNINA-9910639996703321
Carvalho Violeta  
Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022
Materiale a stampa
Lo trovi qui: Univ. Federico II
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Monoclonal Antibodies and Their Functional Fragments in Research, Diagnosis and Therapy
Monoclonal Antibodies and Their Functional Fragments in Research, Diagnosis and Therapy
Autore Ruvo Menotti
Pubbl/distr/stampa Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022
Descrizione fisica 1 electronic resource (278 p.)
Soggetto topico Technology: general issues
Soggetto non controllato porcine deltacoronavirus
nucleocapsid
monoclonal antibodies
neurodegenerative disorders
affibody molecules
blood–brain barrier
receptor-mediated transcytosis
transferrin receptor
AL amyloidosis
CD38
anti-CD38 MoAb
Daratumumab
Isatuximab
myeloma
BCMA
bispecific T-cell engager
antibody-drug conjugates
chimeric antigen receptor T-cells
belantamab mafodotin
idecabtagene vicleucel
JNJ-68284528
Mabs
Antibody-Drug Conjugate
cancer therapy
drug targeting
payload
cross-linking
antibody fragment
Fab
scFv
E. coli
YKL-40
CHI3L1
monoclonal antibody
phage display
lung metastasis
prostate-specific membrane antigen
in vivo imaging
prostate cancer
glutamate carboxypeptidase II
NAALADase
immunization
antibody
protocol
guinea pig
cDNA
chimeric antigen receptor (CAR T)
universal CAR T
modular CAR T
universal immune receptor
CAR adaptor
adoptive immunotherapy
split CAR
bispecific
polyspecificity
pharmacokinetics
solubility
aggregation
viscosity
developability
stability
affinity
specificity
protein engineering
self-association
non-specific binding
immunogenicity
antibody fragments
single chain
amyloid
oligomer
neurotoxicity
NUsc1
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Record Nr. UNINA-9910557613003321
Ruvo Menotti  
Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022
Materiale a stampa
Lo trovi qui: Univ. Federico II
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Nutraceutical, Nutrition Supplements and Human Health
Nutraceutical, Nutrition Supplements and Human Health
Autore Siddiqui Rafat A
Pubbl/distr/stampa Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2020
Descrizione fisica 1 electronic resource (348 p.)
Soggetto topico Research & information: general
Biology, life sciences
Food & society
Soggetto non controllato Lactobacillus salivarius
otitis
probiotic
bacteriocin
prevention
Morus nigra L.
black mulberry
nutraceutical
pharmacological properties
coenzyme Q10 (CoQ10)
bioavailability
intestinal absorption
neuroprotection
fenugreek
protein hydrolysate
antiproliferative
apoptosis
antioxidant
Caco2 cells
catechins
green tea extract
herbal dietary supplements
hepatotoxicity
microbiome
Streptococcus agalactiae
GBS
pregnancy
cachexia
plum
cancer
muscle wasting
myoblasts
protein synthesis
graviola
weight loss
obesity
blood glucose
food composition
metabolic syndrome
natural products
Carica papaya
Bifidobacterium breve M-16V
infant health
clinical efficacy
probiotics
gut microbiota
Autism spectrum disorder
dietary supplements
pediatric
physician communication
frankincense
Boswellia
boswellic acid
lupeolic acid
AKBA
cytokine
breast cancer
pentacyclic triterpenic acid
triterpenoid
chorioallantoic membrane assay
Platycodon grandiflorus root
BMI
body fat mass
abdominal fat area
wild rice
metabolomics
atherosclerosis
LDL-r-KO mice
cytokines
16S rDNA
plasma
feces
proteins
carbohydrates
functional food
curcumin
formulated curcumin
pharmacokinetics
aurora kinase A
hepatocellular carcinoma
Dietary Supplement Label Database
food description
food classification
FoodEx2
quelites
supplementation
arsenic
vitamin K
diet supplement
age-related diseases
vitamin K-dependent proteins
pathological calcification
inflammation
skeletal muscles
Bifidobacterium breve B-3
muscle mass
mitochondria
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Record Nr. UNINA-9910557507803321
Siddiqui Rafat A  
Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2020
Materiale a stampa
Lo trovi qui: Univ. Federico II
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Pharmacogenomics and Personalized Medicine
Pharmacogenomics and Personalized Medicine
Autore Cecchin Erika
Pubbl/distr/stampa Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2020
Descrizione fisica 1 electronic resource (208 p.)
Soggetto topico Medicine
Soggetto non controllato CYP2C9
VKORC1
warfarin
warfarin initiation phase of therapy
INR
pharmacogenetics study
pharmacogenomics
pharmacogenetics
genotype
phenotype
alleles
precision medicine
pharmacotranscriptomics
high-throughput analysis
childhood acute lymphoblastic leukemia
clopidogrel
acenocoumarol
CDSS
implementation
azathioprine
inflammatory bowel disease
glutathione-S transferase
pharmacokinetics
nucleoside analogs
microRNAs
gene expression
drug resistance
AML
cisplatin
nephrotoxicity
kidney injury
genetic polymorphisms
pre-emptive
panel
breast cancer subtype
miRNA
pathway
crosstalk network
precision drugs
ovarian cancer
platinum resistance
focal copy number alterations
whole exome sequencing
personalized medicine
human genetics
pharmacology
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Record Nr. UNINA-9910557287703321
Cecchin Erika  
Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2020
Materiale a stampa
Lo trovi qui: Univ. Federico II
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Precision Medicine : Applied Concepts of Pharmacogenomics in Patients with Various Diseases and Polypharmacy
Precision Medicine : Applied Concepts of Pharmacogenomics in Patients with Various Diseases and Polypharmacy
Autore Turgeon Jacques
Pubbl/distr/stampa Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022
Descrizione fisica 1 electronic resource (170 p.)
Soggetto topico Medicine
Clinical & internal medicine
Soggetto non controllato fibromyalgia (FM)
myalgic encephalomyelitis/chronic fatigue syndrome (ME/CFS)
microRNA
miRNome
pharmacogenomics
pharmacoepigenomics
SM2miR
Pharmaco-miR
repoDB
ME/CFS Common Data Elements (CDEs)
dihydropyrimidine dehydrogenase
DPYD
5-fluorouracil
fluoropyrimidine
therapeutic drug monitoring
orthotopic liver transplant
busulfan
glutathione S-transferase
genetic polymorphism
limited sampling strategy
pharmacokinetics
clinical pharmacogenetics
pharmacogenetic testing
adverse drug reactions
genotype
phenotype
pharmacogene
barriers to pharmacogenetics implementation
Sub-Saharan Africa
chronic low back pain (cLBP)
genetics
personalized treatment
polymorphism
CYP450
tacrolimus
CYP3A5
liver transplant
pharmacogenomic
minority
data collection
drug
biomarker
pharmacogenetics
pharmacogenetic test
personalized medicine
gene expression
infliximab
adalimumab
ulcerative colitis
Crohn disease
inflammatory bowel disease
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Altri titoli varianti Precision Medicine
Record Nr. UNINA-9910585940803321
Turgeon Jacques  
Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022
Materiale a stampa
Lo trovi qui: Univ. Federico II
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Preclinical Evaluation of Lipid-Based Nanosystems
Preclinical Evaluation of Lipid-Based Nanosystems
Autore Silva Ana Catarina
Pubbl/distr/stampa Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021
Descrizione fisica 1 electronic resource (351 p.)
Soggetto topico Technology: general issues
Soggetto non controllato nanostructured lipid carriers (NLC)
formulation optimization
rivastigmine
quality by design (QbD)
nasal route
nose-to-brain
N-alkylisatin
liposome
urokinase plasminogen activator
PAI-2
SerpinB2
breast cancer
liposomes
target delivery nanosystem
FZD10 protein
colon cancer therapy
supersaturation
silica-lipid hybrid
spray drying
lipolysis
lipid-based formulation
fenofibrate
mesoporous silica
oral drug delivery
hyaluronic acid
drug release
light activation
stability
mobility
biocorona
dissolution enhancement
phospholipids
solid dosage forms
porous microparticles
nanoemulsion(s)
phase-behavior
DoE
D-optimal design
vegetable oils
non-ionic surfactants
efavirenz
flaxseed oil
nanostructured lipid carriers
nanocarrier
docohexaenoic acid
neuroprotection
neuroinflammation
fluconazole
Box‒Behnken design
nanotransfersome
ulcer index
zone of inhibition
rheological behavior
ex vivo permeation
nanomedicine
cancer
doxorubicin
melanoma
drug delivery
ultrasound contrast agents
phospholipid coating
ligand distribution
cholesterol
acoustic response
microbubble
lipid phase
dialysis
ammonia
intoxication
cyanocobalamin
vitamin B12
atopic dermatitis
psoriasis
transferosomes
lipid vesicles
skin topical delivery
oligonucleotide
self-emulsifying drug delivery systems
hydrophobic ion pairing
intestinal permeation enhancers
Caco-2 monolayer
clarithromycin
solid lipid nanoparticles
optimization
permeation
pharmacokinetics
follicular targeting
dexamethasone
alopecia areata
lipomers
lipid polymer hybrid nanocapsules
biodistribution
skin
ethyl cellulose
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Record Nr. UNINA-9910557544303321
Silva Ana Catarina  
Basel, Switzerland, : MDPI - Multidisciplinary Digital Publishing Institute, 2021
Materiale a stampa
Lo trovi qui: Univ. Federico II
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Progress and Recent Advances in Solid Organ Transplantation
Progress and Recent Advances in Solid Organ Transplantation
Autore Thongprayoon Charat
Pubbl/distr/stampa Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022
Descrizione fisica 1 electronic resource (188 p.)
Soggetto topico Medicine
Pharmacology
Soggetto non controllato living donation
nephrectomy
hand-assisted laparoscopic nephrectomy
body composition
complications
simultaneous pancreas-kidney transplantation
immunosuppression
graft order
sequence
outcome
survival
kidney transplantation
hydrogen
diarrhea
small intestinal bacterial overgrowth
sickle cell disease
sickle cell
transplantation
outcomes
big data
tacrolimus
metabolism
C/D ratio
cholesterol
dyslipidemia
LDL-C
liver transplantation
hematuria
chronic kidney disease
tocilizumab
clazakizumab
desensitization
anti-HLA alloantibody
post traumatic growth
psychiatric morbidity
network analysis
ESAS
MINI
CPC
DCPR
distress
demoralization
alexithymia
anxiety
antibody-mediated rejection
recurrent primary disease
renal transplantation
pancreas transplantation
cold ischemia time
delayed graft function
Eurotransplant Senior Program
end-stage renal disease
intensive care unit
bioimpedance analysis
drug dosing
lean body mass index
pharmacokinetics
tacrolimus C/D ratio
mineral bone disorder
parathyroidectomy
parathyroid hormone
osteoporosis
bone fractures
Contrast-enhanced ultrasound
kidney perfusion
kidney function
kidney donation
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Record Nr. UNINA-9910576885203321
Thongprayoon Charat  
Basel, : MDPI - Multidisciplinary Digital Publishing Institute, 2022
Materiale a stampa
Lo trovi qui: Univ. Federico II
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Qualitative and Quantitative Analysis of Bioactive Natural Products 2018
Qualitative and Quantitative Analysis of Bioactive Natural Products 2018
Autore Marcotullio Maria Carla
Pubbl/distr/stampa MDPI - Multidisciplinary Digital Publishing Institute, 2019
Descrizione fisica 1 electronic resource (374 p.)
Soggetto non controllato Scorzonera
capsaicinoids
artificial neural network
cerebral ischemia reperfusion injury
antioxidant activity
quality evaluation
chemometrics
secondary metabolites
identification
antioxidant capacity
Moroccan region
volatile compounds
HPLC-Q-Exactive-Orbitrap-MS
quantitative analysis
amino acids content
HPLC-ELSD
antioxidant
autophagy
quantification
sugars
1-triacontanol
hemp seed oil
Alzheimer’s disease
macrodiolides
extraction
recycling preparative high performance liquid chromatography
HPLC methods
GC-MS
Myristica fragrans
Rossa da inverno sel. Rojo Duro onion cultivar
fruit powders
decursin
food traceability
ionic liquids
separation optimisation
Spondias spp
C-glycosylflavone
wine
UPLC-MS
scutellarein
saffron
carotenoids
red cabbage
hydrodistillation
Ginkgo biloba Extract (GBE)
gas chromatography
organic acids
olive leaves
crocins
CBD oil
Bolbostemma paniculatum
UPLC-ESI-MS/MS
geographical origin
HPLC
traditional Chinese medicine decoction
liquid chromatography
bioactive natural compounds
Podospermum
metabolic profiling
SPME-GC/MS
LTQ-Orbitrap
oral administration
UPLC
bioactive compounds
Erigeron breviscapus extract
terrain conditions
nutmeg
antibacterial activity
method validation
ShenFu prescription decoction
chili
decursinol angelate
statistical evaluations
stereoselective and simultaneous analysis
curcuminoids
Talaromyces pinophilus
talarodiolide
HPLC-Q-TOF-MS/MS
Olea europaea L.
triterpenes
chromatogram-bioactivity correlation
essential oil
stability
Staphylococcus aureus
Iris lactea Pall. var. chinensis (Fisch.) Koidz
endothelial function
anthocyanins
HPLC analysis
liquid chromatography-mass spectrometry
nodakenin
turmerone
UHPLC-MS/MS
Quercus acuta leaf
Curcuma longa
UHPLC analysis
ginseng berry extract
geographical variation
qualitative analysis
Sorbus
free radical-scavenging
ginsenosides
flavonoids
biostimulant
GC/MS
terpenes
aleuritolic acid
phenolic compounds
apoptosis
response surface methodology
phenolic acids
pharmacokinetics
mass spectrometry
scutellarin
multivariate statistical analysis
phenolics
MODDE experimental design
proanthocyanidins
UFLC-QQQ-MS
rice
cannabidiol
odor-activity values
UPLC-QTOF-MS
turmeric
decursinol
Formato Materiale a stampa
Livello bibliografico Monografia
Lingua di pubblicazione eng
Record Nr. UNINA-9910346662303321
Marcotullio Maria Carla  
MDPI - Multidisciplinary Digital Publishing Institute, 2019
Materiale a stampa
Lo trovi qui: Univ. Federico II
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