1.

Record Nr.

UNISALENTO991001962459707536

Titolo

Biblia sacra : vulgatae editionis Sixti 5. Pontificis Maximi jussu recognita et Clementis 8. auctoritate edita

Pubbl/distr/stampa

Paris : Garnier, stampa 1922

Edizione

[Nova editio accuratissime emendata a DD. Archiepiscopo parisiensi approvata]

Descrizione fisica

xxviii, 1373 p. ; 20 cm.

Lingua di pubblicazione

Latino

Formato

Materiale a stampa

Livello bibliografico

Monografia

2.

Record Nr.

UNISALENTO991003431109707536

Autore

Seidel Menchi, Silvana

Titolo

Ketzerverfolgung : im 16. und frühen 17. Jahrhundert / in Gemeinschaft mit Hans Rudolf Guggisberg und Bernd Moeller herausgegeben von Silvana Seidel Menchi

Pubbl/distr/stampa

Wiesbaden : Harrassowitz, 1992

ISBN

3447032537

Descrizione fisica

xi, 271 p. ; 23 cm.

Collana

Wolfenbütteler Forschungen ; Bd. 51

Altri autori (Persone)

Guggisberg, Hans R.author

Moeller, Bernd

Soggetti

Heresies, Christian - Storia - Congressi

Heretics, Christian - Congressi

Persecuzioni - Europa - Storia

Lingua di pubblicazione

Inglese

Inglese

Formato

Materiale a stampa

Livello bibliografico

Monografia

Note generali

"Vorträge gehalten anlässlich eines Arbeitsrgesprächs vom 1. bis 5. Oktober 1989 in der Herzog August Bibliothek Wolfenbüttel"--Verso of t.p.



3.

Record Nr.

UNINA9910163348503321

Autore

Rainer Peter

Titolo

Pipeline to battle : an engineer's adventures with the British Eighth army / / Major Peter Rainer

Pubbl/distr/stampa

[Place of publication not identified] : , : Pickle Partners Publishing, , 2013

©1943

ISBN

1-78289-485-3

Descrizione fisica

1 online resource (319 pages)

Disciplina

940.548142

Soggetti

World War, 1939-1945

Lingua di pubblicazione

Inglese

Formato

Materiale a stampa

Livello bibliografico

Monografia



4.

Record Nr.

UNINA9911020074203321

Titolo

Drug bioavailability : estimation of solubility, permeability, absorption and bioavailability

Pubbl/distr/stampa

Weinheim, : Wiley-VCH, c2009

ISBN

9786612307041

9781282307049

1282307045

9783527623860

3527623868

9783527623877

3527623876

Edizione

[2nd, completely rev. ed /]

Descrizione fisica

1 online resource (653 p.)

Collana

Methods and principles in medicinal chemistry ; ; 40

Altri autori (Persone)

WaterbeemdHan van de

TestaBernard

Disciplina

615.19

664.06

Soggetti

Drugs - Bioavailability

Pharmaceutical chemistry

Lingua di pubblicazione

Inglese

Formato

Materiale a stampa

Livello bibliografico

Monografia

Note generali

Description based upon print version of record.

Nota di bibliografia

Includes bibliographical references and index.

Nota di contenuto

Drug Bioavailability: Estimation of Solubility, Permeability, Absorption and Bioavailability; Contents; List of Contributors; Preface; A Personal Foreword; 1 Introduction: The Why and How of Drug Bioavailability Research; 1.1 Dening Bioavailability; 1.1.1 The Biological Context; 1.1.2 A Pharmacokinetic Overview; 1.1.3 Specic Issues; 1.2 Presentation and Layout of the Book; References; Part One Physicochemical Aspects of Drug Dissolution and Solubility; 2 Aqueous Solubility in Drug Discovery Chemistry, DMPK, and Biological Assays; 2.1 Introduction; 2.1.1 Denition of Aqueous Solubility

2.1.2 Aqueous Solubility in Different Phases of Drug Discovery2.2 Aqueous Solubility in Hit Identication; 2.2.1 Aqueous Solubility from DMSO Solutions; 2.2.1.1 Turbidimetric Methods; 2.2.1.2 UV Absorption Methods; 2.2.1.3 Alternative Detection Methodology; 2.2.1.4 Application of DMSO-Based Solubility Assays; 2.3 Aqueous Solubility in



Lead Identication and Lead Optimization; 2.3.1 Dried-Down Solution Methods; 2.3.2 Solubility from Solid; 2.3.3 Thermodynamic Solubility Assays with Solid-State Characterization; 2.3.4 Solubility by Potentiometry

2.3.5 Application of Thermodynamic Solubility Data in LI and LO2.4 Conclusions; References; 3 Gastrointestinal Dissolution and Absorption of Class II Drugs; 3.1 Introduction; 3.2 Drug Absorption and the BCS; 3.3 Class II Drugs; 3.4 GI Physiological Variables Affecting Class II Drug Dissolution; 3.4.1 Bile Salts; 3.4.2 GI pH; 3.4.3 GI Transit; 3.4.4 Drug Particle Size; 3.4.5 Volume Available for Dissolution; 3.5 In Vitro Dissolution Tests for Class II Drugs; 3.5.1 Biorelevant Media; 3.5.2 Dynamic Lipolysis Model; 3.6 BCS-Based FDA Guidelines: Implications for Class II Drugs

3.6.1 Potential of Redening BCS Solubility Class Boundary3.6.2 Biowaiver Extension Potential for Class II Drugs; 3.7 Conclusions; References; 4 In Silico Prediction of Solubility; 4.1 Introduction; 4.2 What Solubility Measures to Model?; 4.3 Is the Data Set Suitable for Modeling?; 4.4 Descriptors and Modeling Methods for Developing Solubility Models; 4.5 Comparing Literature Solubility Models; 4.6 What Is the Inuence of the Domain of Applicability?; 4.7 Can We Tell when Good Predictions Are Made?; 4.8 Conclusions; References

Part Two Physicochemical and Biological Studies of Membrane Permeability and Oral Absorption5 Physicochemical Approaches to Drug Absorption; 5.1 Introduction; 5.2 Physicochemical Properties and Pharmacokinetics; 5.2.1 DMPK; 5.2.2 Lipophilicity, Permeability, and Absorption; 5.2.3 Estimation of Volume of Distribution from Physical Chemistry; 5.2.4 Plasma Protein Binding and Physicochemical Properties; 5.3 Dissolution and Solubility; 5.3.1 Calculated Solubility; 5.4 Ionization (pKa); 5.4.1 Calculated pKa; 5.5 Molecular Size and Shape; 5.5.1 Calculated Size Descriptors; 5.6 Hydrogen Bonding

5.6.1 Calculated Hydrogen-Bonding Descriptors

Sommario/riassunto

The gold standard for industrial research now completely revised in line with current trends in the field, with all contributions extensively updated or rewritten. In 21 chapters readers can benefit from the key working knowledge of today's leading pharmaceutical companies, including Pfizer, AstraZeneca, and Roche. Drug developers from industry and academia present all the factors governing drug bioavailability, complete with practical examples and real-life data. Part I focuses on in vitro and in vivo measurements of physicochemical properties, such as membrane permeability and ioniza