1.

Record Nr.

UNICASUBO2416487

Autore

Vian, Giovanni Maria

Titolo

La donazione di Costantino / Giovanni Maria Vian

Pubbl/distr/stampa

Bologna, : Il mulino, [2004]

ISBN

8815097015

Descrizione fisica

240 p. ; 21 cm.

Collana

L'identità italiana ; 35

Disciplina

262.132

Soggetti

Donazione di Costantino

Lingua di pubblicazione

Italiano

Formato

Materiale a stampa

Livello bibliografico

Monografia

2.

Record Nr.

UNINA9911019428703321

Titolo

Protein kinases as drug targets / / edited by Bert Klebl, Gerhard Muller, and Michael Hamacher

Pubbl/distr/stampa

Weinheim, Germany, : Wiley-VCH, 2011

ISBN

9786613283245

9783527633494

3527633499

9781283283243

1283283247

9783527633470

3527633472

9783527633487

3527633480

Edizione

[2nd ed.]

Descrizione fisica

1 online resource (398 p.)

Collana

Methods and principles in medicinal chemistry ; ; v. 49

Altri autori (Persone)

MullerGerhard

KleblBert

HamacherMichael

Disciplina

615.19

Soggetti

Protein kinases

Drugs - Design



Lingua di pubblicazione

Inglese

Formato

Materiale a stampa

Livello bibliografico

Monografia

Note generali

Description based upon print version of record.

Nota di bibliografia

Includes bibliographical references and index.

Nota di contenuto

pt. 1. Hit finding and profiling for protein kinases : assay development and screening, libraries -- pt. 2. Medicinal chemistry -- pt. 3. Application of kinase inhibitors to therapeutic indication areas.

Sommario/riassunto

This timely guide to kinase inhibitor drug development is the first to cover the entire drug pipeline, from target identification to compound development and clinical application. Edited by the pioneers in the field, on the drug development side this ready reference discusses classical medicinal chemistry approaches as well as current chemical genomics strategies. On the clinical side, both current and future therapeutic application areas for kinase inhibitor drugs are addressed, with a strong focus on oncology drugs.Backed by recent clinical experience with first-generation drugs in the b