1.

Record Nr.

UNINA9910831035503321

Titolo

Mutagenic impurities : strategies for identification and control / / edited by Andrew Teasdale

Pubbl/distr/stampa

Hoboken, New Jersey : , : John Wiley & Sons, Incorporated, , [2022]

©2022

ISBN

1-119-55126-9

1-119-55125-0

1-119-55124-2

Descrizione fisica

1 online resource (547 pages)

Disciplina

576.542

Soggetti

Drugs - Testing

Mutagenicity testing

Lingua di pubblicazione

Inglese

Formato

Materiale a stampa

Livello bibliografico

Monografia

Nota di bibliografia

Includes bibliographical references and index.

Nota di contenuto

Historical perspective on the development of the EMEA Guideline and subsequent ICH M7 Guideline -- ICH M7 -assessment and control of DNA reactive (mutagenic) impurities in pharmaceuticals to limit potential carcinogenic risk -- Control strategies for mutagenic impurities -- Use of structure-activity relationship (SAR) evaluation as a critical tool in the evaluation of the genotoxic potential of impurities -- Evolution of quantitative structure-activity relationships ((Q)SAR) for mutagenicity -- Toxicity testing to understand the mutagenicity of pharmaceutical impurities -- Compound- and class-specific limits for common impurities in pharmaceuticals -- Genotoxic threshold mechanisms and points of departure -- Mutagenic impurities -assessment of fate and control options -- N-nitrosamines -- Conditions potentially leading to the formation of mutagenic impurities -- Strategic approaches to the chromatographic analysis of mutagenic impurities -- Analysis of mutagenic impurities by nuclear magnetic resonance (NMR) spectroscopy -- Addressing the complex problem of degradation-derived mutagenic impurities in drug substances and products.

Sommario/riassunto

"This book examines mutagenic impurities and their impact on the



pharmaceutical industry, following the adoption of the ICH M7 guideline, while focusing on mutagenic impurities from both a toxicological and analytical perspective. The book serves as a primary reference point for anyone faced with addressing the issue of mutagenic impurities, providing readers with a definitive narrative of the guidelines and actual practical solutions to allow them to develop effective control measures"--