1.

Record Nr.

UNINA9910467485103321

Autore

El-Kattan Ayman F.

Titolo

Oral bioavailability assessment : basics and strategies for drug discovery and development / / Ayman F. El-Kattan

Pubbl/distr/stampa

Hoboken, New Jersey : , : Wiley Blackwell, , 2017

©2017

ISBN

1-118-91693-X

1-118-91694-8

1-118-91692-1

Descrizione fisica

1 online resource (455 pages) : illustrations

Collana

Wiley Series on Pharmaceutical Science and Biotechnology: Practices, Applications and Methods

Disciplina

615.1/9

Soggetti

Dental pharmacology

Electronic books.

Lingua di pubblicazione

Inglese

Formato

Materiale a stampa

Livello bibliografico

Monografia

Nota di bibliografia

Includes bibliographical references and index.

Nota di contenuto

Drug pharmacokinetics and toxicokinetics -- GIT anatomy and physiology and drug oral bioavailability : impact of species differences -- Drug routes of excretion -- Physicochemical and biopharmaceutical properties that affect drug absorption of compounds absorbed by passive diffusion -- Physicochemical and biopharmaceutical factors affecting hepatic/intestinal first pass effect -- Impact of intestinal efflux transporters on oral absorption -- Impact of influx transporters on drug -- Extended Clearance Classification System (ECCS) and its utility in predicting clearance rate determining step in drug discovery -- In vitro and in situ approaches to measure intestinal permeability and efflux transporters -- In silico approaches to predict intestinal permeability -- In vivo preclinical approaches to deconvolute the contribution of first pass effect from oral absorption -- In vitro approaches to assess haptic metabolism and first pass effect -- The utility of ECCS as a roadmap to improve oral bioavailability of new molecular entities : industrial perspective.



2.

Record Nr.

UNINA9910305658103321

Titolo

Miglioramento genetico delle piante agrarie / Franco Lorenzetti ... [et al.]

Pubbl/distr/stampa

Milano, : Edagricole, 2018

ISBN

978-88-506-5509-0

Edizione

[[2. ed.]]

Descrizione fisica

XX, 424 p. : ill. ; 26 cm

Disciplina

631.5233

Locazione

FAGBC

NAP11

Collocazione

60 631.523 LORF 2018 BIS

60 631.523 LORF 2018

60 631.523 LORF 2018 TER

631.523 LORF 2018 QUA

631.523 LORF 2018 QUI

631.5233-LOR-1

Lingua di pubblicazione

Italiano

Formato

Materiale a stampa

Livello bibliografico

Monografia

Note generali

Autori dell'edizione precedente:  Franco Lorenzetti, Mario Falcinelli, Fabio Veronesi