1.

Record Nr.

UNINA9910143983503321

Titolo

Drug discovery and development . Volume 2 Drug development [[electronic resource] /] / edited by Mukund S. Chorghade

Pubbl/distr/stampa

Hoboken, N.J., : Wiley-Interscience, c2007

ISBN

1-281-00213-5

9786611002138

0-470-08522-3

0-470-08521-5

Descrizione fisica

1 online resource (401 p.)

Altri autori (Persone)

ChorghadeMukund S (Mukund Shankar)

Disciplina

615.1072

615.19

Soggetti

Drug development

Pharmacology

Lingua di pubblicazione

Inglese

Formato

Materiale a stampa

Livello bibliografico

Monografia

Note generali

Description based upon print version of record.

Nota di bibliografia

Includes bibliographical references and index.

Nota di contenuto

DRUG DISCOVERY AND DEVELOPMENT; CONTENTS; Contributors; Preface; 17 Bioactive Molecules in Medicinal Plants: A Perspective on Their Therapeutic Action; 17.1 Introduction; 17.2 Evolutionary Relationships Among Plants and Humans; 17.3 Traditional Wisdom; 17.4 Unique Libraries for Plants; 17.5 Drugs and Bioactive Molecules from Plants; 17.6 Synergism in Herbal Formulations; 17.7 Interactions Between Modern Drugs and Natural Products; 17.8 Bioavailability and Bioefficacy Enhancers; 17.9 Combination Therapies in Modern Drugs; 17.10 Role of Developments in Technologies and Analytical Tools

17.10.1 Developments in Separation Technologies17.10.2 Developments in Combined Techniques and Advanced Technologies; 17.10.3 Molecular Farming and Bioengineering of Medicinal Plants; 17.10.4 High-Throughput Screening of Natural Products; 17.11 Herbal Medicine: The Best Possible Route to Health Care; References; 18 Natural Products as an Inspiration for the Discovery of New High-Throughput Chemical Synthesis Tools; 18.1 Introduction; 18.2 Solid-Supported Reagents as Tools in Natural Product Synthesis; 18.3 Multistep Use of Supported Reagents in Natural Product Synthesis; 18.4



Conclusions

References19 Insulin Sensitizers: Emerging Therapeutics; 19.1 Introduction; 19.2 Therapeutic Interventions; 19.3 Discovery of Insulin Sensitizers; 19.4 Journey Toward New Drugs; 19.5 Conclusions; References; 20 Criteria for Industrial Readiness of Chiral Catalysis Technology for the Synthesis of Pharmaceuticals; 20.1 Introduction; 20.2 Criteria for Technology Readiness; 20.3 Examples of Industrially Ready Chiral Catalytic Technologies and Their Application; 20.3.1 Lipase Bioresolution: Ethyl 3-Amino-3-Phenylpropionate; 20.3.2 Aminoacylase Bioresolution of N-Acylamino Acids

20.3.3 Asymmetric Hydrogenation of Prochiral Olefins by Rhodium-DuPhos Catalysts20.3.4 Asymmetric Hydrogenation of Prochiral Ketones by Ruthenium-Biphosphine-Diamine Catalysts; 20.3.5 Asymmetric Hydroformylation with Rhodium-Phosphite Catalysts; 20.3.6 Asymmetric Allylic Substitution with Palladium-Based Catalysts; 20.4 How Industrially Ready Technology Can Deliver Commercial Advantages; 20.5 Conclusions; References; 21 Enantioselective Synthesis of Propargyl Alcohols as Multifunctional Synthons; 21.1 Introduction; 21.2 Asymmetric Reduction of Prochiral α, β-Alkynyl Ketones

21.3 Addition of Acetylenic Anion to Carbonyl Carbon21.4 Desymmetrization and Enzymatic Strategies for Chiral Propargyl Alcohol Synthesis; 21.5 β-Elimination Strategy and Miscellaneous Approaches; 21.6 Conclusions; References; 22 Carbohydrates: From Chirons to Mimics; 22.1 Introduction; 22.2 Synthetic Strategies for C-Glycosides; 22.3 Synthetic Strategies for Carbon-Linked Disaccharides and Pseudosaccharides; References; 23 Meeting the Challenges of Process Development and Scale-up of Active Pharmaceutical Ingredients; 23.1 Introduction; 23.1.1 Drug Development in the Pharmaceutical Industry

23.1.2 Challenges in Developing and Scaling Up Chemical Processes

Sommario/riassunto

From first principles to real-world applications-here is the first comprehensive guide to drug discovery and development Modern drug discovery and development require the collaborative efforts of specialists in a broadarray of scientific, technical, and business disciplines-from biochemistry to molecular biology, organic chemistry to medicinal chemistry, pharmacology to marketing. Yet surprisingly, until now, there were no authoritative references offering a complete, fully integrated picture of the process. The only comprehensive guide of its kind, this groundbreaking two-volume re



2.

Record Nr.

UNINA9910713433903321

Autore

Stamey Timothy C.

Titolo

Frequency and duration of flooding of Grove Creek near Kenansville, North Carolina, for present and proposed restored channel conditions / / by T.C. Stamey

Pubbl/distr/stampa

Raleigh, North Carolina : , : U.S. Geological Survey, , 1985

Descrizione fisica

1 online resource (v, 52 pages) : illustrations, maps

Collana

Water-resources investigations report ; ; 85-4298

Soggetti

Flood forecasting - North Carolina - Kenansville Region

Floods - North Carolina - Kenansville Region

River channels - North Carolina

Flood forecasting

Floods

Lingua di pubblicazione

Inglese

Formato

Materiale a stampa

Livello bibliografico

Monografia

Note generali

"Prepared in cooperation with North Carolina Department of Human Resources."

Nota di bibliografia

Includes bibliographical references (pages 29).



3.

Record Nr.

UNINA9910792166103321

Autore

Freire Paulo <1921-1997.>

Titolo

Pedagogy of Solidarity [[electronic resource]]

Pubbl/distr/stampa

Walnut Creek, : Left Coast Press, 2014

ISBN

1-315-42280-8

1-315-42279-4

1-315-42281-6

1-61132-966-3

Descrizione fisica

1 online resource (124 p.)

Collana

Qualitative Inquiry & Social Justice

Altri autori (Persone)

Araújo FreireAna María <1933->

OliveiraWalter Ferreira de

Disciplina

370.115

Soggetti

Community and school

Critical pedagogy

EDUCATION / Philosophy & Social Aspects

POLITICAL SCIENCE / Political Freedom & Security / Human Rights

Popular education

SOCIAL SCIENCE / Methodology

Lingua di pubblicazione

Inglese

Formato

Materiale a stampa

Livello bibliografico

Monografia

Note generali

Description based upon print version of record.

Nota di contenuto

Contents; Foreword - Memory's Hope: In the Shadow of Paulo Freire's Presence - Henry A. Giroux; Chapter 1. Introduction to Pedagogy of Solidarity - Walter Ferreira de Oliveira; Chapter 2. Pedagogy of Solidarity - Paulo Freire; Chapter 3. Pedagogy of Solidarity: A Dialogue - Paulo Freire; Chapter 4. For a Pedagogy of Solidarity - Walter Ferreira de Oliveira; Chapter 5. Testimony of Difference and the Right to Discuss Difference - Ana Maria Araújo Freire; Chapter 6. The Importance of Pedagogy of Solidarity - Norman K. Denzin; Afterword - Re-imaging Freire Beyond Methods - Donaldo Macedo; Index

About the Authors

Sommario/riassunto

Famous Brazilian educational and social theorist Paulo Freire presents his ideas on the importance of community solidarity in moving toward social justice in schools and society. In a set of talks and interviews shortly before his death, Freire addresses issues not often highlighted



in his work, such as globalization, post-modern fatalism, and the qualities of educators for the 21st century. His illuminating comments are supplemented with commentaries by other well-known scholars, such as Ana Maria Araujo Freire, Norman Denzin, Henry Giroux, and Donaldo Macedo.